Design, synthesis, and pharmacological evaluation of a novel series of pyridopyrazine-1,6-dione γ-secretase modulators.
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| Title: | Design, synthesis, and pharmacological evaluation of a novel series of pyridopyrazine-1,6-dione γ-secretase modulators. |
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| Authors: | Pettersson M; Pfizer Worldwide Research & Development , 610 Main Street, Cambridge, Massachusetts 02139, United States., Johnson DS, Subramanyam C, Bales KR, am Ende CW, Fish BA, Green ME, Kauffman GW, Mullins PB, Navaratnam T, Sakya SM, Stiff CM, Tran TP, Xie L, Zhang L, Pustilnik LR, Vetelino BC, Wood KM, Pozdnyakov N, Verhoest PR, O'Donnell CJ |
| Source: | Journal of medicinal chemistry [J Med Chem] 2014 Feb 13; Vol. 57 (3), pp. 1046-62. Date of Electronic Publication: 2014 Jan 28. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 24428186 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=24428186 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/jm401782h Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1046 Titles: – TitleFull: Design, synthesis, and pharmacological evaluation of a novel series of pyridopyrazine-1,6-dione γ-secretase modulators. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Pettersson M – PersonEntity: Name: NameFull: Johnson DS – PersonEntity: Name: NameFull: Subramanyam C – PersonEntity: Name: NameFull: Bales KR – PersonEntity: Name: NameFull: am Ende CW – PersonEntity: Name: NameFull: Fish BA – PersonEntity: Name: NameFull: Green ME – PersonEntity: Name: NameFull: Kauffman GW – PersonEntity: Name: NameFull: Mullins PB – PersonEntity: Name: NameFull: Navaratnam T – PersonEntity: Name: NameFull: Sakya SM – PersonEntity: Name: NameFull: Stiff CM – PersonEntity: Name: NameFull: Tran TP – PersonEntity: Name: NameFull: Xie L – PersonEntity: Name: NameFull: Zhang L – PersonEntity: Name: NameFull: Pustilnik LR – PersonEntity: Name: NameFull: Vetelino BC – PersonEntity: Name: NameFull: Wood KM – PersonEntity: Name: NameFull: Pozdnyakov N – PersonEntity: Name: NameFull: Verhoest PR – PersonEntity: Name: NameFull: O'Donnell CJ IsPartOfRelationships: – BibEntity: Dates: – D: 13 M: 02 Text: 2014 Feb 13 Type: published Y: 2014 Identifiers: – Type: issn-electronic Value: 1520-4804 Numbering: – Type: volume Value: 57 – Type: issue Value: 3 Titles: – TitleFull: Journal of medicinal chemistry Type: main |
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