Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening.

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Title: Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening.
Authors: Yang B; Oncology Innovative Medicine Unit, AstraZeneca R&D Boston , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States., Lamb ML, Zhang T, Hennessy EJ, Grewal G, Sha L, Zambrowski M, Block MH, Dowling JE, Su N, Wu J, Deegan T, Mikule K, Wang W, Kaspera R, Chuaqui C, Chen H
Source: Journal of medicinal chemistry [J Med Chem] 2014 Dec 11; Vol. 57 (23), pp. 9958-70. Date of Electronic Publication: 2014 Dec 02.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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An: 25458601
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  Data: Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening.
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  Data: <searchLink fieldCode="AU" term="%22Yang+B%22">Yang B</searchLink>; Oncology Innovative Medicine Unit, AstraZeneca R&D Boston , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Lamb+ML%22">Lamb ML</searchLink><br /><searchLink fieldCode="AU" term="%22Zhang+T%22">Zhang T</searchLink><br /><searchLink fieldCode="AU" term="%22Hennessy+EJ%22">Hennessy EJ</searchLink><br /><searchLink fieldCode="AU" term="%22Grewal+G%22">Grewal G</searchLink><br /><searchLink fieldCode="AU" term="%22Sha+L%22">Sha L</searchLink><br /><searchLink fieldCode="AU" term="%22Zambrowski+M%22">Zambrowski M</searchLink><br /><searchLink fieldCode="AU" term="%22Block+MH%22">Block MH</searchLink><br /><searchLink fieldCode="AU" term="%22Dowling+JE%22">Dowling JE</searchLink><br /><searchLink fieldCode="AU" term="%22Su+N%22">Su N</searchLink><br /><searchLink fieldCode="AU" term="%22Wu+J%22">Wu J</searchLink><br /><searchLink fieldCode="AU" term="%22Deegan+T%22">Deegan T</searchLink><br /><searchLink fieldCode="AU" term="%22Mikule+K%22">Mikule K</searchLink><br /><searchLink fieldCode="AU" term="%22Wang+W%22">Wang W</searchLink><br /><searchLink fieldCode="AU" term="%22Kaspera+R%22">Kaspera R</searchLink><br /><searchLink fieldCode="AU" term="%22Chuaqui+C%22">Chuaqui C</searchLink><br /><searchLink fieldCode="AU" term="%22Chen+H%22">Chen H</searchLink>
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2014 Dec 11; Vol. 57 (23), pp. 9958-70. <i>Date of Electronic Publication: </i>2014 Dec 02.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
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        Value: 10.1021/jm501179r
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      – Code: eng
        Text: English
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        StartPage: 9958
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      – TitleFull: Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening.
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              Text: 2014 Dec 11
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              Value: 57
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              Value: 23
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