Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening.
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| Title: | Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening. |
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| Authors: | Yang B; Oncology Innovative Medicine Unit, AstraZeneca R&D Boston , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States., Lamb ML, Zhang T, Hennessy EJ, Grewal G, Sha L, Zambrowski M, Block MH, Dowling JE, Su N, Wu J, Deegan T, Mikule K, Wang W, Kaspera R, Chuaqui C, Chen H |
| Source: | Journal of medicinal chemistry [J Med Chem] 2014 Dec 11; Vol. 57 (23), pp. 9958-70. Date of Electronic Publication: 2014 Dec 02. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 25458601 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Yang+B%22">Yang B</searchLink>; Oncology Innovative Medicine Unit, AstraZeneca R&D Boston , 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States.<br /><searchLink fieldCode="AU" term="%22Lamb+ML%22">Lamb ML</searchLink><br /><searchLink fieldCode="AU" term="%22Zhang+T%22">Zhang T</searchLink><br /><searchLink fieldCode="AU" term="%22Hennessy+EJ%22">Hennessy EJ</searchLink><br /><searchLink fieldCode="AU" term="%22Grewal+G%22">Grewal G</searchLink><br /><searchLink fieldCode="AU" term="%22Sha+L%22">Sha L</searchLink><br /><searchLink fieldCode="AU" term="%22Zambrowski+M%22">Zambrowski M</searchLink><br /><searchLink fieldCode="AU" term="%22Block+MH%22">Block MH</searchLink><br /><searchLink fieldCode="AU" term="%22Dowling+JE%22">Dowling JE</searchLink><br /><searchLink fieldCode="AU" term="%22Su+N%22">Su N</searchLink><br /><searchLink fieldCode="AU" term="%22Wu+J%22">Wu J</searchLink><br /><searchLink fieldCode="AU" term="%22Deegan+T%22">Deegan T</searchLink><br /><searchLink fieldCode="AU" term="%22Mikule+K%22">Mikule K</searchLink><br /><searchLink fieldCode="AU" term="%22Wang+W%22">Wang W</searchLink><br /><searchLink fieldCode="AU" term="%22Kaspera+R%22">Kaspera R</searchLink><br /><searchLink fieldCode="AU" term="%22Chuaqui+C%22">Chuaqui C</searchLink><br /><searchLink fieldCode="AU" term="%22Chen+H%22">Chen H</searchLink> – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2014 Dec 11; Vol. 57 (23), pp. 9958-70. <i>Date of Electronic Publication: </i>2014 Dec 02. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=25458601 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/jm501179r Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 9958 Titles: – TitleFull: Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Yang B – PersonEntity: Name: NameFull: Lamb ML – PersonEntity: Name: NameFull: Zhang T – PersonEntity: Name: NameFull: Hennessy EJ – PersonEntity: Name: NameFull: Grewal G – PersonEntity: Name: NameFull: Sha L – PersonEntity: Name: NameFull: Zambrowski M – PersonEntity: Name: NameFull: Block MH – PersonEntity: Name: NameFull: Dowling JE – PersonEntity: Name: NameFull: Su N – PersonEntity: Name: NameFull: Wu J – PersonEntity: Name: NameFull: Deegan T – PersonEntity: Name: NameFull: Mikule K – PersonEntity: Name: NameFull: Wang W – PersonEntity: Name: NameFull: Kaspera R – PersonEntity: Name: NameFull: Chuaqui C – PersonEntity: Name: NameFull: Chen H IsPartOfRelationships: – BibEntity: Dates: – D: 11 M: 12 Text: 2014 Dec 11 Type: published Y: 2014 Identifiers: – Type: issn-electronic Value: 1520-4804 Numbering: – Type: volume Value: 57 – Type: issue Value: 23 Titles: – TitleFull: Journal of medicinal chemistry Type: main |
| ResultId | 1 |