Structure-based drug design identifies polythiophenes as antiprion compounds.

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Title: Structure-based drug design identifies polythiophenes as antiprion compounds.
Authors: Herrmann US; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Schütz AK; Physical Chemistry, Eidgenössische Technische Hochschule (ETH) Zürich, 8093 Zürich, Switzerland., Shirani H; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden., Huang D; Department of Biochemistry, University of Zürich, 8057 Zürich, Switzerland., Saban D; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Nuvolone M; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Li B; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Ballmer B; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Åslund AK; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden., Mason JJ; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden., Rushing E; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Budka H; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland., Nyström S; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden., Hammarström P; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden., Böckmann A; Institut de Biologie et Chimie des Protéines, UMR 5086 CNRS/Université de Lyon 1, 69367 Lyon, France., Caflisch A; Department of Biochemistry, University of Zürich, 8057 Zürich, Switzerland., Meier BH; Physical Chemistry, Eidgenössische Technische Hochschule (ETH) Zürich, 8093 Zürich, Switzerland., Nilsson KP; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden., Hornemann S; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland. adriano.aguzzi@usz.ch simone.hornemann@usz.ch., Aguzzi A; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland. adriano.aguzzi@usz.ch simone.hornemann@usz.ch.
Source: Science translational medicine [Sci Transl Med] 2015 Aug 05; Vol. 7 (299), pp. 299ra123.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Association for the Advancement of Science Country of Publication: United States NLM ID: 101505086 Publication Model: Print Cited Medium: Internet ISSN: 1946-6242 (Electronic) Linking ISSN: 19466234 NLM ISO Abbreviation: Sci Transl Med Subsets: MEDLINE
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  Data: Structure-based drug design identifies polythiophenes as antiprion compounds.
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  Data: <searchLink fieldCode="AU" term="%22Herrmann+US%22">Herrmann US</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Schütz+AK%22">Schütz AK</searchLink>; Physical Chemistry, Eidgenössische Technische Hochschule (ETH) Zürich, 8093 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Shirani+H%22">Shirani H</searchLink>; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden.<br /><searchLink fieldCode="AU" term="%22Huang+D%22">Huang D</searchLink>; Department of Biochemistry, University of Zürich, 8057 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Saban+D%22">Saban D</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Nuvolone+M%22">Nuvolone M</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Li+B%22">Li B</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Ballmer+B%22">Ballmer B</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Åslund+AK%22">Åslund AK</searchLink>; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden.<br /><searchLink fieldCode="AU" term="%22Mason+JJ%22">Mason JJ</searchLink>; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden.<br /><searchLink fieldCode="AU" term="%22Rushing+E%22">Rushing E</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Budka+H%22">Budka H</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Nyström+S%22">Nyström S</searchLink>; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden.<br /><searchLink fieldCode="AU" term="%22Hammarström+P%22">Hammarström P</searchLink>; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden.<br /><searchLink fieldCode="AU" term="%22Böckmann+A%22">Böckmann A</searchLink>; Institut de Biologie et Chimie des Protéines, UMR 5086 CNRS/Université de Lyon 1, 69367 Lyon, France.<br /><searchLink fieldCode="AU" term="%22Caflisch+A%22">Caflisch A</searchLink>; Department of Biochemistry, University of Zürich, 8057 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Meier+BH%22">Meier BH</searchLink>; Physical Chemistry, Eidgenössische Technische Hochschule (ETH) Zürich, 8093 Zürich, Switzerland.<br /><searchLink fieldCode="AU" term="%22Nilsson+KP%22">Nilsson KP</searchLink>; Department of Physics, Chemistry and Biology (IFM), Linköping University, 58183 Linköping, Sweden.<br /><searchLink fieldCode="AU" term="%22Hornemann+S%22">Hornemann S</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland. adriano.aguzzi@usz.ch simone.hornemann@usz.ch.<br /><searchLink fieldCode="AU" term="%22Aguzzi+A%22">Aguzzi A</searchLink>; Institute of Neuropathology, University Hospital of Zürich, University of Zürich, 8091 Zürich, Switzerland. adriano.aguzzi@usz.ch simone.hornemann@usz.ch.
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