Benzimidazole analogs as WTA biosynthesis inhibitors targeting methicillin resistant Staphylococcus aureus.

Saved in:
Bibliographic Details
Title: Benzimidazole analogs as WTA biosynthesis inhibitors targeting methicillin resistant Staphylococcus aureus.
Authors: Yang SW; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States. Electronic address: shu-wei.yang@merck.com., Pan J; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Yang C; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Labroli M; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Pan W; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Caldwell J; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Ha S; Structure Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Koseoglu S; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Xiao JC; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Mayhood T; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Sheth PR; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Garlisi CG; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Wu J; Pharmacokinetics PPDM, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Lee SH; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Wang H; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Tan CM; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Roemer T; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Su J; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2016 Oct 01; Vol. 26 (19), pp. 4743-4747. Date of Electronic Publication: 2016 Aug 16.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1464-3405
DOI:10.1016/j.bmcl.2016.08.036