Benzimidazole analogs as WTA biosynthesis inhibitors targeting methicillin resistant Staphylococcus aureus.
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| Title: | Benzimidazole analogs as WTA biosynthesis inhibitors targeting methicillin resistant Staphylococcus aureus. |
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| Authors: | Yang SW; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States. Electronic address: shu-wei.yang@merck.com., Pan J; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Yang C; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Labroli M; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Pan W; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Caldwell J; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Ha S; Structure Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Koseoglu S; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Xiao JC; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Mayhood T; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Sheth PR; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Garlisi CG; In Vitro Pharmacology Group, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Wu J; Pharmacokinetics PPDM, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Lee SH; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Wang H; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Tan CM; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Roemer T; Infectious Disease, Merck Research Laboratory, Kenilworth, NJ 07033, United States., Su J; Discovery Chemistry, Merck Research Laboratory, Kenilworth, NJ 07033, United States. |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2016 Oct 01; Vol. 26 (19), pp. 4743-4747. Date of Electronic Publication: 2016 Aug 16. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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