Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder.

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Bibliographic Details
Title: Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladder.
Authors: Harper BH; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States. Electronic address: bart_harper@merck.com., Wang L; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Zhu C; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Kar NF; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Li B; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Moyes CR; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Goble SD; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Costa M; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Dingley K; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Di Salvo J; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Ha SN; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Hurley A; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Li X; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Miller RR; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Nagabukuro H; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Salituro GM; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Smith S; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Struthers M; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Hale JJ; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Edmondson SD; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States., Berger R; Merck & Co., Inc., 126 E. Lincoln Ave., Rahway, NJ 07065, United States.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Feb 15; Vol. 27 (4), pp. 1094-1098. Date of Electronic Publication: 2016 Dec 11.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1464-3405
DOI:10.1016/j.bmcl.2016.12.033