Identification of novel TACE inhibitors compatible with topical application.

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Title: Identification of novel TACE inhibitors compatible with topical application.
Authors: Ouvry G; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: gilles.ouvry@galderma.com., Berton Y; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bhurruth-Alcor Y; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bonnary L; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bouix-Peter C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bouquet K; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bourotte M; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Chambon S; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Comino C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Deprez B; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Duvert D; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Duvert G; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hacini-Rachinel F; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Harris CS; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Luzy AP; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Mathieu A; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Millois C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pascau J; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pinto A; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Polge G; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Reitz A; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Reversé K; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Rosignoli C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Taquet N; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hennequin LF; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
Source: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2017 Apr 15; Vol. 27 (8), pp. 1848-1853. Date of Electronic Publication: 2017 Feb 20.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Identification of novel TACE inhibitors compatible with topical application.
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  Data: <searchLink fieldCode="AU" term="%22Ouvry+G%22">Ouvry G</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: gilles.ouvry@galderma.com.<br /><searchLink fieldCode="AU" term="%22Berton+Y%22">Berton Y</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Bhurruth-Alcor+Y%22">Bhurruth-Alcor Y</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Bonnary+L%22">Bonnary L</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Bouix-Peter+C%22">Bouix-Peter C</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Bouquet+K%22">Bouquet K</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Bourotte+M%22">Bourotte M</searchLink>; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France.<br /><searchLink fieldCode="AU" term="%22Chambon+S%22">Chambon S</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Comino+C%22">Comino C</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Deprez+B%22">Deprez B</searchLink>; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France.<br /><searchLink fieldCode="AU" term="%22Duvert+D%22">Duvert D</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Duvert+G%22">Duvert G</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Hacini-Rachinel+F%22">Hacini-Rachinel F</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Harris+CS%22">Harris CS</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Luzy+AP%22">Luzy AP</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Mathieu+A%22">Mathieu A</searchLink>; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France.<br /><searchLink fieldCode="AU" term="%22Millois+C%22">Millois C</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pascau+J%22">Pascau J</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pinto+A%22">Pinto A</searchLink>; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France.<br /><searchLink fieldCode="AU" term="%22Polge+G%22">Polge G</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Reitz+A%22">Reitz A</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Reversé+K%22">Reversé K</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Rosignoli+C%22">Rosignoli C</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Taquet+N%22">Taquet N</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Hennequin+LF%22">Hennequin LF</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
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