Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.

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Title: Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.
Authors: Fadeyi OO; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Hoth LR; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Choi C; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Feng X; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Gopalsamy A; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States., Hett EC; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States., Kyne RE Jr; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Robinson RP; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Jones LH; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States.
Source: ACS chemical biology [ACS Chem Biol] 2017 Aug 18; Vol. 12 (8), pp. 2015-2020. Date of Electronic Publication: 2017 Jul 20.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
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  Data: Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.
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  Data: <searchLink fieldCode="AU" term="%22Fadeyi+OO%22">Fadeyi OO</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Hoth+LR%22">Hoth LR</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Choi+C%22">Choi C</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Feng+X%22">Feng X</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Gopalsamy+A%22">Gopalsamy A</searchLink>; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Hett+EC%22">Hett EC</searchLink>; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Kyne+RE+Jr%22">Kyne RE Jr</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Robinson+RP%22">Robinson RP</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Jones+LH%22">Jones LH</searchLink>; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States.
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  Data: <searchLink fieldCode="JN" term="%22101282906%22">ACS chemical biology</searchLink> [ACS Chem Biol] 2017 Aug 18; Vol. 12 (8), pp. 2015-2020. <i>Date of Electronic Publication: </i>2017 Jul 20.
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        Value: 10.1021/acschembio.7b00403
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        StartPage: 2015
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      – TitleFull: Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.
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              Text: 2017 Aug 18
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