Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.
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| Title: | Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue. |
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| Authors: | Fadeyi OO; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Hoth LR; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Choi C; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Feng X; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Gopalsamy A; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States., Hett EC; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States., Kyne RE Jr; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Robinson RP; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Jones LH; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States. |
| Source: | ACS chemical biology [ACS Chem Biol] 2017 Aug 18; Vol. 12 (8), pp. 2015-2020. Date of Electronic Publication: 2017 Jul 20. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 28718624 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Fadeyi+OO%22">Fadeyi OO</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Hoth+LR%22">Hoth LR</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Choi+C%22">Choi C</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Feng+X%22">Feng X</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Gopalsamy+A%22">Gopalsamy A</searchLink>; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Hett+EC%22">Hett EC</searchLink>; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Kyne+RE+Jr%22">Kyne RE Jr</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Robinson+RP%22">Robinson RP</searchLink>; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Jones+LH%22">Jones LH</searchLink>; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101282906%22">ACS chemical biology</searchLink> [ACS Chem Biol] 2017 Aug 18; Vol. 12 (8), pp. 2015-2020. <i>Date of Electronic Publication: </i>2017 Jul 20. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101282906 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1554-8937 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2215548929%22">15548929 </searchLink><i>NLM ISO Abbreviation: </i>ACS Chem Biol <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=28718624 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acschembio.7b00403 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 2015 Titles: – TitleFull: Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Fadeyi OO – PersonEntity: Name: NameFull: Hoth LR – PersonEntity: Name: NameFull: Choi C – PersonEntity: Name: NameFull: Feng X – PersonEntity: Name: NameFull: Gopalsamy A – PersonEntity: Name: NameFull: Hett EC – PersonEntity: Name: NameFull: Kyne RE Jr – PersonEntity: Name: NameFull: Robinson RP – PersonEntity: Name: NameFull: Jones LH IsPartOfRelationships: – BibEntity: Dates: – D: 18 M: 08 Text: 2017 Aug 18 Type: published Y: 2017 Identifiers: – Type: issn-electronic Value: 1554-8937 Numbering: – Type: volume Value: 12 – Type: issue Value: 8 Titles: – TitleFull: ACS chemical biology Type: main |
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