Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue.
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| Title: | Covalent Enzyme Inhibition through Fluorosulfate Modification of a Noncatalytic Serine Residue. |
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| Authors: | Fadeyi OO; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Hoth LR; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Choi C; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Feng X; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Gopalsamy A; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States., Hett EC; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States., Kyne RE Jr; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Robinson RP; Medicine Design, Pfizer Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Jones LH; Medicine Design, Pfizer Inc. , 610 Main Street, Cambridge, Massachusetts 02139, United States. |
| Source: | ACS chemical biology [ACS Chem Biol] 2017 Aug 18; Vol. 12 (8), pp. 2015-2020. Date of Electronic Publication: 2017 Jul 20. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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