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Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis.

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Title: Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis.
Authors: Boiteau JG; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: jean-guy.boiteau@galderma.com., Ouvry G; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: gilles.ouvry@galderma.com., Arlabosse JM; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Astri S; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Beillard A; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bhurruth-Alcor Y; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bonnary L; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bouix-Peter C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bouquet K; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bourotte M; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Cardinaud I; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Comino C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Deprez B; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Duvert D; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Féret A; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hacini-Rachinel F; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Harris CS; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Luzy AP; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Mathieu A; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Millois C; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Orsini N; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pascau J; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pinto A; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France., Piwnica D; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Polge G; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Reitz A; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Reversé K; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Rodeville N; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Rossio P; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Spiesse D; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Tabet S; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Taquet N; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Tomas L; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Vial E; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hennequin LF; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
Source: Bioorganic & medicinal chemistry [Bioorg Med Chem] 2018 Feb 15; Vol. 26 (4), pp. 945-956. Date of Electronic Publication: 2017 Aug 02.
Publication Type: Journal Article
Journal Info: Publisher: Elsevier Science Country of Publication: England NLM ID: 9413298 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3391 (Electronic) Linking ISSN: 09680896 NLM ISO Abbreviation: Bioorg Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis.
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  Data: <searchLink fieldCode="AU" term="%22Boiteau+JG%22">Boiteau JG</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: jean-guy.boiteau@galderma.com.<br /><searchLink fieldCode="AU" term="%22Ouvry+G%22">Ouvry G</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France. 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Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France.<br /><searchLink fieldCode="AU" term="%22Millois+C%22">Millois C</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Orsini+N%22">Orsini N</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pascau+J%22">Pascau J</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pinto+A%22">Pinto A</searchLink>; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177 - Drugs and Molecules for Living Systems, F-59000 Lille, France.<br /><searchLink fieldCode="AU" term="%22Piwnica+D%22">Piwnica D</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Polge+G%22">Polge G</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Reitz+A%22">Reitz A</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Reversé+K%22">Reversé K</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Rodeville+N%22">Rodeville N</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Rossio+P%22">Rossio P</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Spiesse+D%22">Spiesse D</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Tabet+S%22">Tabet S</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Taquet+N%22">Taquet N</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Tomas+L%22">Tomas L</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Vial+E%22">Vial E</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Hennequin+LF%22">Hennequin LF</searchLink>; Nestlé Skin Health R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
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