Design, Synthesis, and Biological Activity of 1,2,3-Triazolobenzodiazepine BET Bromodomain Inhibitors.
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| Title: | Design, Synthesis, and Biological Activity of 1,2,3-Triazolobenzodiazepine BET Bromodomain Inhibitors. |
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| Authors: | Sharp PP; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Garnier JM; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Hatfaludi T; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Xu Z; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Segal D; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Jarman KE; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Jousset H; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Garnham A; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Feutrill JT; Synthesis MedChem, 399 Royal Parade, Parkville, VIC 3052, Australia., Cuzzupe A; Synthesis MedChem, 399 Royal Parade, Parkville, VIC 3052, Australia., Hall P; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Taylor S; St. Vincent's Institute of Medical Research and Department of Medicine, St Vincent's Hospital, University of Melbourne, Fitzroy, VIC 3052, Australia., Walkley CR; St. Vincent's Institute of Medical Research and Department of Medicine, St Vincent's Hospital, University of Melbourne, Fitzroy, VIC 3052, Australia., Tyler D; Cancer Research Division, Peter MacCallum Cancer Centre, Melbourne, VIC 3000, Australia., Dawson MA; Cancer Research Division, Peter MacCallum Cancer Centre, Melbourne, VIC 3000, Australia.; Department of Haematology, Peter MacCallum Cancer Centre, Melbourne, VIC 3000, Australia.; Sir Peter MacCallum Department of Oncology, The University of Melbourne, East Melbourne, VIC 3002, Australia., Czabotar P; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Wilks AF; Synthesis MedChem, 399 Royal Parade, Parkville, VIC 3052, Australia., Glaser S; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Huang DCS; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia., Burns CJ; Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, VIC 3052, Australia.; Department of Medical Biology, The University of Melbourne, Melbourne, VIC 3010, Australia.; School of Chemistry, The Bio21 Institute, The University of Melbourne, Melbourne, VIC 3010, Australia. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2017 Nov 14; Vol. 8 (12), pp. 1298-1303. Date of Electronic Publication: 2017 Nov 14 (Print Publication: 2017). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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