Discovery of a Stress-Activated Protein Kinase Inhibitor for Lymphatic Filariasis.

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Title: Discovery of a Stress-Activated Protein Kinase Inhibitor for Lymphatic Filariasis.
Authors: Tummalapalli SR; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Bhat R; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Chojnowski A; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Prorok M; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Kreiss T; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Goldberg R; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Canan S; Celgene Global Health, Celgene San Diego, 10300 Campus Point Drive, San Diego, California 92121, United States., Hawryluk N; Celgene Global Health, Celgene San Diego, 10300 Campus Point Drive, San Diego, California 92121, United States., Mortensen D; Celgene Global Health, Celgene San Diego, 10300 Campus Point Drive, San Diego, California 92121, United States., Khetani V; Celgene Global Health, 86 Morris Avenue, Summit, New Jersey 07901, United States., Zeldis J; Celgene Global Health, 86 Morris Avenue, Summit, New Jersey 07901, United States., Siekierka JJ; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States., Rotella DP; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2018 Feb 09; Vol. 9 (3), pp. 210-214. Date of Electronic Publication: 2018 Feb 09 (Print Publication: 2018).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
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  Data: <searchLink fieldCode="AU" term="%22Tummalapalli+SR%22">Tummalapalli SR</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Bhat+R%22">Bhat R</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Chojnowski+A%22">Chojnowski A</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Prorok+M%22">Prorok M</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Kreiss+T%22">Kreiss T</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Goldberg+R%22">Goldberg R</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Canan+S%22">Canan S</searchLink>; Celgene Global Health, Celgene San Diego, 10300 Campus Point Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Hawryluk+N%22">Hawryluk N</searchLink>; Celgene Global Health, Celgene San Diego, 10300 Campus Point Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Mortensen+D%22">Mortensen D</searchLink>; Celgene Global Health, Celgene San Diego, 10300 Campus Point Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Khetani+V%22">Khetani V</searchLink>; Celgene Global Health, 86 Morris Avenue, Summit, New Jersey 07901, United States.<br /><searchLink fieldCode="AU" term="%22Zeldis+J%22">Zeldis J</searchLink>; Celgene Global Health, 86 Morris Avenue, Summit, New Jersey 07901, United States.<br /><searchLink fieldCode="AU" term="%22Siekierka+JJ%22">Siekierka JJ</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.<br /><searchLink fieldCode="AU" term="%22Rotella+DP%22">Rotella DP</searchLink>; Sokol Institute for Pharmaceutical Life Sciences and Department of Chemistry and Biochemistry, Montclair State University, Montclair, New Jersey 07043, United States.
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  Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2018 Feb 09; Vol. 9 (3), pp. 210-214. <i>Date of Electronic Publication: </i>2018 Feb 09 (<i>Print Publication: </i>2018).
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        Value: 10.1021/acsmedchemlett.7b00477
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