Sulfoximines as potent RORγ inverse agonists.
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| Title: | Sulfoximines as potent RORγ inverse agonists. |
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| Authors: | Ouvry G; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: gilles.ouvry@galderma.com., Bihl F; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Bouix-Peter C; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Christin O; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Defoin-Platel C; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Deret S; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Feret C; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Froude D; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hacini-Rachinel F; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Harris CS; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hervouet C; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Lafitte G; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Luzy AP; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Musicki B; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Orfila D; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Parnet V; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pascau C; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pascau J; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Pierre R; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Raffin C; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Rossio P; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Spiesse D; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Taquet N; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Thoreau E; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Vatinel R; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Vial E; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France., Hennequin LF; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France. |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2018 May 01; Vol. 28 (8), pp. 1269-1273. Date of Electronic Publication: 2018 Mar 17. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 29571573 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Sulfoximines as potent RORγ inverse agonists. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Ouvry+G%22">Ouvry G</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France. Electronic address: gilles.ouvry@galderma.com.<br /><searchLink fieldCode="AU" term="%22Bihl+F%22">Bihl F</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Bouix-Peter+C%22">Bouix-Peter C</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Christin+O%22">Christin O</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Defoin-Platel+C%22">Defoin-Platel C</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Deret+S%22">Deret S</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Feret+C%22">Feret C</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Froude+D%22">Froude D</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Hacini-Rachinel+F%22">Hacini-Rachinel F</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Harris+CS%22">Harris CS</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Hervouet+C%22">Hervouet C</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Lafitte+G%22">Lafitte G</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Luzy+AP%22">Luzy AP</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Musicki+B%22">Musicki B</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Orfila+D%22">Orfila D</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Parnet+V%22">Parnet V</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pascau+C%22">Pascau C</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pascau+J%22">Pascau J</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Pierre+R%22">Pierre R</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Raffin+C%22">Raffin C</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Rossio+P%22">Rossio P</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Spiesse+D%22">Spiesse D</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Taquet+N%22">Taquet N</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Thoreau+E%22">Thoreau E</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Vatinel+R%22">Vatinel R</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Vial+E%22">Vial E</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France.<br /><searchLink fieldCode="AU" term="%22Hennequin+LF%22">Hennequin LF</searchLink>; Nestlé Skin Health, Les Templiers 2400 Route des Colles, 06410 Biot, France. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2018 May 01; Vol. 28 (8), pp. 1269-1273. <i>Date of Electronic Publication: </i>2018 Mar 17. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
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| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2018.03.041 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1269 Titles: – TitleFull: Sulfoximines as potent RORγ inverse agonists. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Ouvry G – PersonEntity: Name: NameFull: Bihl F – PersonEntity: Name: NameFull: Bouix-Peter C – PersonEntity: Name: NameFull: Christin O – PersonEntity: Name: NameFull: Defoin-Platel C – PersonEntity: Name: NameFull: Deret S – PersonEntity: Name: NameFull: Feret C – PersonEntity: Name: NameFull: Froude D – PersonEntity: Name: NameFull: Hacini-Rachinel F – PersonEntity: Name: NameFull: Harris CS – PersonEntity: Name: NameFull: Hervouet C – PersonEntity: Name: NameFull: Lafitte G – PersonEntity: Name: NameFull: Luzy AP – PersonEntity: Name: NameFull: Musicki B – PersonEntity: Name: NameFull: Orfila D – PersonEntity: Name: NameFull: Parnet V – PersonEntity: Name: NameFull: Pascau C – PersonEntity: Name: NameFull: Pascau J – PersonEntity: Name: NameFull: Pierre R – PersonEntity: Name: NameFull: Raffin C – PersonEntity: Name: NameFull: Rossio P – PersonEntity: Name: NameFull: Spiesse D – PersonEntity: Name: NameFull: Taquet N – PersonEntity: Name: NameFull: Thoreau E – PersonEntity: Name: NameFull: Vatinel R – PersonEntity: Name: NameFull: Vial E – PersonEntity: Name: NameFull: Hennequin LF IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 05 Text: 2018 May 01 Type: published Y: 2018 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 28 – Type: issue Value: 8 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
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