Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1).
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| Title: | Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1). |
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| Authors: | Filipski KJ; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Sammons MF; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Bhattacharya SK; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Panteleev J; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States., Brown JA; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States., Loria PM; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States., Boehm M; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Smith AC; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States., Shavnya A; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States., Conn EL; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States., Song K; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Weng Y; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Facemire C; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Jüppner H; Endocrine Unit and Pediatric Nephrology Unit, Thier 10, Massachusetts General Hospital and Harvard Medical School, 50 Blossom Street, Boston, Massachusetts 02114, United States., Clerin V; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2018 Apr 12; Vol. 9 (5), pp. 440-445. Date of Electronic Publication: 2018 Apr 12 (Print Publication: 2018). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 29795756 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1). – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Filipski+KJ%22">Filipski KJ</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Sammons+MF%22">Sammons MF</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Bhattacharya+SK%22">Bhattacharya SK</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Panteleev+J%22">Panteleev J</searchLink>; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Brown+JA%22">Brown JA</searchLink>; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Loria+PM%22">Loria PM</searchLink>; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Boehm+M%22">Boehm M</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Smith+AC%22">Smith AC</searchLink>; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Shavnya+A%22">Shavnya A</searchLink>; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Conn+EL%22">Conn EL</searchLink>; Pfizer Worldwide Research & Development, 558 Eastern Point Road, Groton, Connecticut 06340, United States.<br /><searchLink fieldCode="AU" term="%22Song+K%22">Song K</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Weng+Y%22">Weng Y</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Facemire+C%22">Facemire C</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States.<br /><searchLink fieldCode="AU" term="%22Jüppner+H%22">Jüppner H</searchLink>; Endocrine Unit and Pediatric Nephrology Unit, Thier 10, Massachusetts General Hospital and Harvard Medical School, 50 Blossom Street, Boston, Massachusetts 02114, United States.<br /><searchLink fieldCode="AU" term="%22Clerin+V%22">Clerin V</searchLink>; Pfizer Worldwide Research & Development, 1 Portland Street, Cambridge, Massachusetts 02139, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2018 Apr 12; Vol. 9 (5), pp. 440-445. <i>Date of Electronic Publication: </i>2018 Apr 12 (<i>Print Publication: </i>2018). – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=29795756 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acsmedchemlett.8b00013 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 440 Titles: – TitleFull: Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1). Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Filipski KJ – PersonEntity: Name: NameFull: Sammons MF – PersonEntity: Name: NameFull: Bhattacharya SK – PersonEntity: Name: NameFull: Panteleev J – PersonEntity: Name: NameFull: Brown JA – PersonEntity: Name: NameFull: Loria PM – PersonEntity: Name: NameFull: Boehm M – PersonEntity: Name: NameFull: Smith AC – PersonEntity: Name: NameFull: Shavnya A – PersonEntity: Name: NameFull: Conn EL – PersonEntity: Name: NameFull: Song K – PersonEntity: Name: NameFull: Weng Y – PersonEntity: Name: NameFull: Facemire C – PersonEntity: Name: NameFull: Jüppner H – PersonEntity: Name: NameFull: Clerin V IsPartOfRelationships: – BibEntity: Dates: – D: 12 M: 04 Text: 2018 Apr 12 Type: published Y: 2018 Identifiers: – Type: issn-print Value: 1948-5875 Numbering: – Type: volume Value: 9 – Type: issue Value: 5 Titles: – TitleFull: ACS medicinal chemistry letters Type: main |
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