Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties.

Saved in:
Bibliographic Details
Title: Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties.
Authors: Santora VJ; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Almos TA; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Barido R; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Basinger J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Bellows CL; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Bookser BC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Breitenbucher JG; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Broadbent NJ; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Cabebe C; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chai CK; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chen M; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chow S; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chung M; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Crickard L; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Danks AM; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Freestone GC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Gitnick D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Gupta V; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Hoffmaster C; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Hudson AR; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Kaplan AP; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Kennedy MR; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Lee D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Limberis J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Ly K; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Mak CC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Masatsugu B; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Morse AC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Na J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Neul D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Nikpur J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Peters M; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Petroski RE; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Renick J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Sebring K; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Sevidal S; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Tabatabaei A; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Wen J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Yan Y; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Yoder ZW; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Zook D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.
Source: Journal of medicinal chemistry [J Med Chem] 2018 Jul 26; Vol. 61 (14), pp. 6018-6033. Date of Electronic Publication: 2018 Jul 11.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 29886732
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Santora+VJ%22">Santora VJ</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Almos+TA%22">Almos TA</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Barido+R%22">Barido R</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Basinger+J%22">Basinger J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Bellows+CL%22">Bellows CL</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Bookser+BC%22">Bookser BC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Breitenbucher+JG%22">Breitenbucher JG</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Broadbent+NJ%22">Broadbent NJ</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Cabebe+C%22">Cabebe C</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chai+CK%22">Chai CK</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chen+M%22">Chen M</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chow+S%22">Chow S</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chung+M%22">Chung M</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Crickard+L%22">Crickard L</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Danks+AM%22">Danks AM</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Freestone+GC%22">Freestone GC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Gitnick+D%22">Gitnick D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Gupta+V%22">Gupta V</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Hoffmaster+C%22">Hoffmaster C</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Hudson+AR%22">Hudson AR</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Kaplan+AP%22">Kaplan AP</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Kennedy+MR%22">Kennedy MR</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Lee+D%22">Lee D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Limberis+J%22">Limberis J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Ly+K%22">Ly K</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Mak+CC%22">Mak CC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Masatsugu+B%22">Masatsugu B</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Morse+AC%22">Morse AC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Na+J%22">Na J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Neul+D%22">Neul D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Nikpur+J%22">Nikpur J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Peters+M%22">Peters M</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Petroski+RE%22">Petroski RE</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Renick+J%22">Renick J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Sebring+K%22">Sebring K</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Sevidal+S%22">Sevidal S</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Tabatabaei+A%22">Tabatabaei A</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Wen+J%22">Wen J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Yan+Y%22">Yan Y</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Yoder+ZW%22">Yoder ZW</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Zook+D%22">Zook D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2018 Jul 26; Vol. 61 (14), pp. 6018-6033. <i>Date of Electronic Publication: </i>2018 Jul 11.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=29886732
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1021/acs.jmedchem.8b00372
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 6018
    Titles:
      – TitleFull: Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Santora VJ
      – PersonEntity:
          Name:
            NameFull: Almos TA
      – PersonEntity:
          Name:
            NameFull: Barido R
      – PersonEntity:
          Name:
            NameFull: Basinger J
      – PersonEntity:
          Name:
            NameFull: Bellows CL
      – PersonEntity:
          Name:
            NameFull: Bookser BC
      – PersonEntity:
          Name:
            NameFull: Breitenbucher JG
      – PersonEntity:
          Name:
            NameFull: Broadbent NJ
      – PersonEntity:
          Name:
            NameFull: Cabebe C
      – PersonEntity:
          Name:
            NameFull: Chai CK
      – PersonEntity:
          Name:
            NameFull: Chen M
      – PersonEntity:
          Name:
            NameFull: Chow S
      – PersonEntity:
          Name:
            NameFull: Chung M
      – PersonEntity:
          Name:
            NameFull: Crickard L
      – PersonEntity:
          Name:
            NameFull: Danks AM
      – PersonEntity:
          Name:
            NameFull: Freestone GC
      – PersonEntity:
          Name:
            NameFull: Gitnick D
      – PersonEntity:
          Name:
            NameFull: Gupta V
      – PersonEntity:
          Name:
            NameFull: Hoffmaster C
      – PersonEntity:
          Name:
            NameFull: Hudson AR
      – PersonEntity:
          Name:
            NameFull: Kaplan AP
      – PersonEntity:
          Name:
            NameFull: Kennedy MR
      – PersonEntity:
          Name:
            NameFull: Lee D
      – PersonEntity:
          Name:
            NameFull: Limberis J
      – PersonEntity:
          Name:
            NameFull: Ly K
      – PersonEntity:
          Name:
            NameFull: Mak CC
      – PersonEntity:
          Name:
            NameFull: Masatsugu B
      – PersonEntity:
          Name:
            NameFull: Morse AC
      – PersonEntity:
          Name:
            NameFull: Na J
      – PersonEntity:
          Name:
            NameFull: Neul D
      – PersonEntity:
          Name:
            NameFull: Nikpur J
      – PersonEntity:
          Name:
            NameFull: Peters M
      – PersonEntity:
          Name:
            NameFull: Petroski RE
      – PersonEntity:
          Name:
            NameFull: Renick J
      – PersonEntity:
          Name:
            NameFull: Sebring K
      – PersonEntity:
          Name:
            NameFull: Sevidal S
      – PersonEntity:
          Name:
            NameFull: Tabatabaei A
      – PersonEntity:
          Name:
            NameFull: Wen J
      – PersonEntity:
          Name:
            NameFull: Yan Y
      – PersonEntity:
          Name:
            NameFull: Yoder ZW
      – PersonEntity:
          Name:
            NameFull: Zook D
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 26
              M: 07
              Text: 2018 Jul 26
              Type: published
              Y: 2018
          Identifiers:
            – Type: issn-electronic
              Value: 1520-4804
          Numbering:
            – Type: volume
              Value: 61
            – Type: issue
              Value: 14
          Titles:
            – TitleFull: Journal of medicinal chemistry
              Type: main
ResultId 1