Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties.
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| Title: | Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties. |
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| Authors: | Santora VJ; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Almos TA; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Barido R; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Basinger J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Bellows CL; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Bookser BC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Breitenbucher JG; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Broadbent NJ; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Cabebe C; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chai CK; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chen M; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chow S; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Chung M; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Crickard L; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Danks AM; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Freestone GC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Gitnick D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Gupta V; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Hoffmaster C; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Hudson AR; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Kaplan AP; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Kennedy MR; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Lee D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Limberis J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Ly K; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Mak CC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Masatsugu B; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Morse AC; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Na J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Neul D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Nikpur J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Peters M; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Petroski RE; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Renick J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Sebring K; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Sevidal S; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Tabatabaei A; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Wen J; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Yan Y; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Yoder ZW; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States., Zook D; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States. |
| Source: | Journal of medicinal chemistry [J Med Chem] 2018 Jul 26; Vol. 61 (14), pp. 6018-6033. Date of Electronic Publication: 2018 Jul 11. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 29886732 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Santora+VJ%22">Santora VJ</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Almos+TA%22">Almos TA</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Barido+R%22">Barido R</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Basinger+J%22">Basinger J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Bellows+CL%22">Bellows CL</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Bookser+BC%22">Bookser BC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Breitenbucher+JG%22">Breitenbucher JG</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Broadbent+NJ%22">Broadbent NJ</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Cabebe+C%22">Cabebe C</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chai+CK%22">Chai CK</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chen+M%22">Chen M</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chow+S%22">Chow S</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Chung+M%22">Chung M</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Crickard+L%22">Crickard L</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Danks+AM%22">Danks AM</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Freestone+GC%22">Freestone GC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Gitnick+D%22">Gitnick D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Gupta+V%22">Gupta V</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Hoffmaster+C%22">Hoffmaster C</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Hudson+AR%22">Hudson AR</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Kaplan+AP%22">Kaplan AP</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Kennedy+MR%22">Kennedy MR</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Lee+D%22">Lee D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Limberis+J%22">Limberis J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Ly+K%22">Ly K</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Mak+CC%22">Mak CC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Masatsugu+B%22">Masatsugu B</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Morse+AC%22">Morse AC</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Na+J%22">Na J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Neul+D%22">Neul D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Nikpur+J%22">Nikpur J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Peters+M%22">Peters M</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Petroski+RE%22">Petroski RE</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Renick+J%22">Renick J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Sebring+K%22">Sebring K</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Sevidal+S%22">Sevidal S</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Tabatabaei+A%22">Tabatabaei A</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Wen+J%22">Wen J</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Yan+Y%22">Yan Y</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Yoder+ZW%22">Yoder ZW</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States.<br /><searchLink fieldCode="AU" term="%22Zook+D%22">Zook D</searchLink>; Dart NeuroScience LLC , 12278 Scripps Summit Drive , San Diego , California 92121 , United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2018 Jul 26; Vol. 61 (14), pp. 6018-6033. <i>Date of Electronic Publication: </i>2018 Jul 11. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE |
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| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acs.jmedchem.8b00372 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 6018 Titles: – TitleFull: Design and Synthesis of Novel and Selective Glycine Transporter-1 (GlyT1) Inhibitors with Memory Enhancing Properties. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Santora VJ – PersonEntity: Name: NameFull: Almos TA – PersonEntity: Name: NameFull: Barido R – PersonEntity: Name: NameFull: Basinger J – PersonEntity: Name: NameFull: Bellows CL – PersonEntity: Name: NameFull: Bookser BC – PersonEntity: Name: NameFull: Breitenbucher JG – PersonEntity: Name: NameFull: Broadbent NJ – PersonEntity: Name: NameFull: Cabebe C – PersonEntity: Name: NameFull: Chai CK – PersonEntity: Name: NameFull: Chen M – PersonEntity: Name: NameFull: Chow S – PersonEntity: Name: NameFull: Chung M – PersonEntity: Name: NameFull: Crickard L – PersonEntity: Name: NameFull: Danks AM – PersonEntity: Name: NameFull: Freestone GC – PersonEntity: Name: NameFull: Gitnick D – PersonEntity: Name: NameFull: Gupta V – PersonEntity: Name: NameFull: Hoffmaster C – PersonEntity: Name: NameFull: Hudson AR – PersonEntity: Name: NameFull: Kaplan AP – PersonEntity: Name: NameFull: Kennedy MR – PersonEntity: Name: NameFull: Lee D – PersonEntity: Name: NameFull: Limberis J – PersonEntity: Name: NameFull: Ly K – PersonEntity: Name: NameFull: Mak CC – PersonEntity: Name: NameFull: Masatsugu B – PersonEntity: Name: NameFull: Morse AC – PersonEntity: Name: NameFull: Na J – PersonEntity: Name: NameFull: Neul D – PersonEntity: Name: NameFull: Nikpur J – PersonEntity: Name: NameFull: Peters M – PersonEntity: Name: NameFull: Petroski RE – PersonEntity: Name: NameFull: Renick J – PersonEntity: Name: NameFull: Sebring K – PersonEntity: Name: NameFull: Sevidal S – PersonEntity: Name: NameFull: Tabatabaei A – PersonEntity: Name: NameFull: Wen J – PersonEntity: Name: NameFull: Yan Y – PersonEntity: Name: NameFull: Yoder ZW – PersonEntity: Name: NameFull: Zook D IsPartOfRelationships: – BibEntity: Dates: – D: 26 M: 07 Text: 2018 Jul 26 Type: published Y: 2018 Identifiers: – Type: issn-electronic Value: 1520-4804 Numbering: – Type: volume Value: 61 – Type: issue Value: 14 Titles: – TitleFull: Journal of medicinal chemistry Type: main |
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