TPT sulfonate, a single, oral dose schistosomicidal prodrug: In vivo efficacy, disposition and metabolic profiling.
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| Title: | TPT sulfonate, a single, oral dose schistosomicidal prodrug: In vivo efficacy, disposition and metabolic profiling. |
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| Authors: | Wolfe AR; Department of Bioengineering and Therapeutic Sciences, University of California San Francisco, 533 Parnassus Ave, San Francisco, CA, 94143, USA; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA., Neitz RJ; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pharmaceutical Chemistry, University of California, 1700 4th St, San Francisco, CA, 94158, USA., Burlingame M; Department of Pharmaceutical Chemistry, University of California, 1700 4th St, San Francisco, CA, 94158, USA., Suzuki BM; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pathology, University of California, 1700 4th St, San Francisco, CA, 94158, USA., Lim KC; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pathology, University of California, 1700 4th St, San Francisco, CA, 94158, USA., Scheideler M; Human First Therapeutics LLC, 9600 Dewitt Drive, Ste 1, Silver Spring, MD, 20910, USA., Nelson DL; Pro-Rectory of Research and Graduate Study, Federal University of the Valleys of Jequitinhonha and Mucuri, 39100-000, Diamantina, MG, Brazil., Benet LZ; Department of Bioengineering and Therapeutic Sciences, University of California San Francisco, 533 Parnassus Ave, San Francisco, CA, 94143, USA; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA., Caffrey CR; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pathology, University of California, 1700 4th St, San Francisco, CA, 94158, USA. Electronic address: ccaffrey@ucsd.edu. |
| Source: | International journal for parasitology. Drugs and drug resistance [Int J Parasitol Drugs Drug Resist] 2018 Dec; Vol. 8 (3), pp. 571-586. Date of Electronic Publication: 2018 Nov 20. |
| Publication Type: | Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: Elsevier Country of Publication: Netherlands NLM ID: 101576715 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2211-3207 (Electronic) Linking ISSN: 22113207 NLM ISO Abbreviation: Int J Parasitol Drugs Drug Resist Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 30503203 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: TPT sulfonate, a single, oral dose schistosomicidal prodrug: In vivo efficacy, disposition and metabolic profiling. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Wolfe+AR%22">Wolfe AR</searchLink>; Department of Bioengineering and Therapeutic Sciences, University of California San Francisco, 533 Parnassus Ave, San Francisco, CA, 94143, USA; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA.<br /><searchLink fieldCode="AU" term="%22Neitz+RJ%22">Neitz RJ</searchLink>; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pharmaceutical Chemistry, University of California, 1700 4th St, San Francisco, CA, 94158, USA.<br /><searchLink fieldCode="AU" term="%22Burlingame+M%22">Burlingame M</searchLink>; Department of Pharmaceutical Chemistry, University of California, 1700 4th St, San Francisco, CA, 94158, USA.<br /><searchLink fieldCode="AU" term="%22Suzuki+BM%22">Suzuki BM</searchLink>; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pathology, University of California, 1700 4th St, San Francisco, CA, 94158, USA.<br /><searchLink fieldCode="AU" term="%22Lim+KC%22">Lim KC</searchLink>; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pathology, University of California, 1700 4th St, San Francisco, CA, 94158, USA.<br /><searchLink fieldCode="AU" term="%22Scheideler+M%22">Scheideler M</searchLink>; Human First Therapeutics LLC, 9600 Dewitt Drive, Ste 1, Silver Spring, MD, 20910, USA.<br /><searchLink fieldCode="AU" term="%22Nelson+DL%22">Nelson DL</searchLink>; Pro-Rectory of Research and Graduate Study, Federal University of the Valleys of Jequitinhonha and Mucuri, 39100-000, Diamantina, MG, Brazil.<br /><searchLink fieldCode="AU" term="%22Benet+LZ%22">Benet LZ</searchLink>; Department of Bioengineering and Therapeutic Sciences, University of California San Francisco, 533 Parnassus Ave, San Francisco, CA, 94143, USA; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA.<br /><searchLink fieldCode="AU" term="%22Caffrey+CR%22">Caffrey CR</searchLink>; Center for Discovery and Innovation in Parasitic Diseases, University of California, 1700 4th St, San Francisco, CA, 94158, USA; Department of Pathology, University of California, 1700 4th St, San Francisco, CA, 94158, USA. Electronic address: ccaffrey@ucsd.edu. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101576715%22">International journal for parasitology. Drugs and drug resistance</searchLink> [Int J Parasitol Drugs Drug Resist] 2018 Dec; Vol. 8 (3), pp. 571-586. <i>Date of Electronic Publication: </i>2018 Nov 20. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>Netherlands <i>NLM ID: </i>101576715 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2211-3207 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2222113207%22">22113207 </searchLink><i>NLM ISO Abbreviation: </i>Int J Parasitol Drugs Drug Resist <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=30503203 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.ijpddr.2018.10.004 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 571 Titles: – TitleFull: TPT sulfonate, a single, oral dose schistosomicidal prodrug: In vivo efficacy, disposition and metabolic profiling. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Wolfe AR – PersonEntity: Name: NameFull: Neitz RJ – PersonEntity: Name: NameFull: Burlingame M – PersonEntity: Name: NameFull: Suzuki BM – PersonEntity: Name: NameFull: Lim KC – PersonEntity: Name: NameFull: Scheideler M – PersonEntity: Name: NameFull: Nelson DL – PersonEntity: Name: NameFull: Benet LZ – PersonEntity: Name: NameFull: Caffrey CR IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 12 Text: 2018 Dec Type: published Y: 2018 Identifiers: – Type: issn-electronic Value: 2211-3207 Numbering: – Type: volume Value: 8 – Type: issue Value: 3 Titles: – TitleFull: International journal for parasitology. Drugs and drug resistance Type: main |
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