Functional characterization of 27 CYP3A4 protein variants to metabolize regorafenib in vitro.

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Title: Functional characterization of 27 CYP3A4 protein variants to metabolize regorafenib in vitro.
Authors: Li YH; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China., Lin QM; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China., Pang NH; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China., Zhang XD; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China., Huang HL; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China., Cai JP; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China., Hu GX; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.
Source: Basic & clinical pharmacology & toxicology [Basic Clin Pharmacol Toxicol] 2019 Oct; Vol. 125 (4), pp. 337-344. Date of Electronic Publication: 2019 Jun 18.
Publication Type: Journal Article
Journal Info: Publisher: Blackwell Country of Publication: England NLM ID: 101208422 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1742-7843 (Electronic) Linking ISSN: 17427835 NLM ISO Abbreviation: Basic Clin Pharmacol Toxicol Subsets: MEDLINE
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  Data: Functional characterization of 27 CYP3A4 protein variants to metabolize regorafenib in vitro.
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  Data: <searchLink fieldCode="AU" term="%22Li+YH%22">Li YH</searchLink>; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.<br /><searchLink fieldCode="AU" term="%22Lin+QM%22">Lin QM</searchLink>; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.<br /><searchLink fieldCode="AU" term="%22Pang+NH%22">Pang NH</searchLink>; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.<br /><searchLink fieldCode="AU" term="%22Zhang+XD%22">Zhang XD</searchLink>; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.<br /><searchLink fieldCode="AU" term="%22Huang+HL%22">Huang HL</searchLink>; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.<br /><searchLink fieldCode="AU" term="%22Cai+JP%22">Cai JP</searchLink>; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Hu+GX%22">Hu GX</searchLink>; Department of Pharmacology, School of Pharmacy, Wenzhou Medical University, Wenzhou, China.
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  Data: <searchLink fieldCode="JN" term="%22101208422%22">Basic & clinical pharmacology & toxicology</searchLink> [Basic Clin Pharmacol Toxicol] 2019 Oct; Vol. 125 (4), pp. 337-344. <i>Date of Electronic Publication: </i>2019 Jun 18.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Blackwell%22">Blackwell </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101208422 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1742-7843 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2217427835%22">17427835 </searchLink><i>NLM ISO Abbreviation: </i>Basic Clin Pharmacol Toxicol <i>Subsets: </i>MEDLINE
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        Value: 10.1111/bcpt.13246
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      – TitleFull: Functional characterization of 27 CYP3A4 protein variants to metabolize regorafenib in vitro.
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              Text: 2019 Oct
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