A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation.

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Title: A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation.
Authors: Sammons RM, Perry NA, Li Y; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States.; Department of Drug Discovery & Biomedical Sciences , University of South Carolina , Columbia , South Carolina 29208 , United States., Cho EJ, Piserchio A; Department of Chemistry and Biochemistry , The City College of New York , New York , New York 10031 , United States., Zamora-Olivares DP, Ghose R; Department of Chemistry and Biochemistry , The City College of New York , New York , New York 10031 , United States., Kaoud TS; Department of Medicinal Chemistry, Faculty of Pharmacy , Minia University , 61519 Minia , Egypt., Debevec G; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States., Bartholomeusz C, Gurevich VV, Iverson TM, Giulianotti M; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States., Houghten RA; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States., Dalby KN
Source: ACS chemical biology [ACS Chem Biol] 2019 Jun 21; Vol. 14 (6), pp. 1183-1194. Date of Electronic Publication: 2019 May 13.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation.
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  Data: <searchLink fieldCode="AU" term="%22Sammons+RM%22">Sammons RM</searchLink><br /><searchLink fieldCode="AU" term="%22Perry+NA%22">Perry NA</searchLink><br /><searchLink fieldCode="AU" term="%22Li+Y%22">Li Y</searchLink>; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States.; Department of Drug Discovery & Biomedical Sciences , University of South Carolina , Columbia , South Carolina 29208 , United States.<br /><searchLink fieldCode="AU" term="%22Cho+EJ%22">Cho EJ</searchLink><br /><searchLink fieldCode="AU" term="%22Piserchio+A%22">Piserchio A</searchLink>; Department of Chemistry and Biochemistry , The City College of New York , New York , New York 10031 , United States.<br /><searchLink fieldCode="AU" term="%22Zamora-Olivares+DP%22">Zamora-Olivares DP</searchLink><br /><searchLink fieldCode="AU" term="%22Ghose+R%22">Ghose R</searchLink>; Department of Chemistry and Biochemistry , The City College of New York , New York , New York 10031 , United States.<br /><searchLink fieldCode="AU" term="%22Kaoud+TS%22">Kaoud TS</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy , Minia University , 61519 Minia , Egypt.<br /><searchLink fieldCode="AU" term="%22Debevec+G%22">Debevec G</searchLink>; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States.<br /><searchLink fieldCode="AU" term="%22Bartholomeusz+C%22">Bartholomeusz C</searchLink><br /><searchLink fieldCode="AU" term="%22Gurevich+VV%22">Gurevich VV</searchLink><br /><searchLink fieldCode="AU" term="%22Iverson+TM%22">Iverson TM</searchLink><br /><searchLink fieldCode="AU" term="%22Giulianotti+M%22">Giulianotti M</searchLink>; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States.<br /><searchLink fieldCode="AU" term="%22Houghten+RA%22">Houghten RA</searchLink>; Torrey Pines Institute for Molecular Studies , Port St. Lucie , Florida 34987 , United States.<br /><searchLink fieldCode="AU" term="%22Dalby+KN%22">Dalby KN</searchLink>
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  Data: <searchLink fieldCode="JN" term="%22101282906%22">ACS chemical biology</searchLink> [ACS Chem Biol] 2019 Jun 21; Vol. 14 (6), pp. 1183-1194. <i>Date of Electronic Publication: </i>2019 May 13.
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  Data: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101282906 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1554-8937 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2215548929%22">15548929 </searchLink><i>NLM ISO Abbreviation: </i>ACS Chem Biol <i>Subsets: </i>MEDLINE
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        Value: 10.1021/acschembio.9b00093
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        Text: English
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              Text: 2019 Jun 21
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