Functional characterization of 27 CYP3A4 variants on macitentan metabolism in vitro.

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Title: Functional characterization of 27 CYP3A4 variants on macitentan metabolism in vitro.
Authors: Li YH; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Lu XR; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Lin QM; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Huang HL; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Liang XL; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Cai JP; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China., Cui J; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China., Hu GX; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.
Source: The Journal of pharmacy and pharmacology [J Pharm Pharmacol] 2019 Nov; Vol. 71 (11), pp. 1677-1683. Date of Electronic Publication: 2019 Aug 22.
Publication Type: Journal Article
Journal Info: Publisher: Oxford University Press Country of Publication: England NLM ID: 0376363 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2042-7158 (Electronic) Linking ISSN: 00223573 NLM ISO Abbreviation: J Pharm Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:2042-7158
DOI:10.1111/jphp.13153