Functional characterization of 27 CYP3A4 variants on macitentan metabolism in vitro.

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Title: Functional characterization of 27 CYP3A4 variants on macitentan metabolism in vitro.
Authors: Li YH; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Lu XR; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Lin QM; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Huang HL; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Liang XL; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China., Cai JP; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China., Cui J; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China., Hu GX; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.
Source: The Journal of pharmacy and pharmacology [J Pharm Pharmacol] 2019 Nov; Vol. 71 (11), pp. 1677-1683. Date of Electronic Publication: 2019 Aug 22.
Publication Type: Journal Article
Journal Info: Publisher: Oxford University Press Country of Publication: England NLM ID: 0376363 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2042-7158 (Electronic) Linking ISSN: 00223573 NLM ISO Abbreviation: J Pharm Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Functional characterization of 27 CYP3A4 variants on macitentan metabolism in vitro.
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  Data: <searchLink fieldCode="AU" term="%22Li+YH%22">Li YH</searchLink>; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.<br /><searchLink fieldCode="AU" term="%22Lu+XR%22">Lu XR</searchLink>; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.<br /><searchLink fieldCode="AU" term="%22Lin+QM%22">Lin QM</searchLink>; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.<br /><searchLink fieldCode="AU" term="%22Huang+HL%22">Huang HL</searchLink>; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.<br /><searchLink fieldCode="AU" term="%22Liang+XL%22">Liang XL</searchLink>; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.<br /><searchLink fieldCode="AU" term="%22Cai+JP%22">Cai JP</searchLink>; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Cui+J%22">Cui J</searchLink>; The Key Laboratory of Geriatrics, Beijing Hospital and Beijing Institute of Geriatrics, Ministry of Health, Beijing, China.<br /><searchLink fieldCode="AU" term="%22Hu+GX%22">Hu GX</searchLink>; School of Pharmaceutical Sciences, Wenzhou Medical University, Wenzhou, Zhejiang, China.
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        Value: 10.1111/jphp.13153
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      – TitleFull: Functional characterization of 27 CYP3A4 variants on macitentan metabolism in vitro.
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              Text: 2019 Nov
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              Y: 2019
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