Activation of the GLP-1 receptor by a non-peptidic agonist.

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Title: Activation of the GLP-1 receptor by a non-peptidic agonist.
Authors: Zhao P; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Liang YL; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Belousoff MJ; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Deganutti G; School of Biological Sciences, University of Essex, Colchester, UK., Fletcher MM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Willard FS; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA., Bell MG; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA., Christe ME; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA., Sloop KW; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA., Inoue A; Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Miyagi, Japan., Truong TT; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Clydesdale L; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Furness SGB; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Christopoulos A; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia., Wang MW; The National Center for Drug Screening and CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China.; School of Pharmacy, Fudan University, Shanghai, China., Miller LJ; Mayo Clinic, Scottsdale, AZ, USA., Reynolds CA; School of Biological Sciences, University of Essex, Colchester, UK., Danev R; Graduate School of Medicine, University of Tokyo, Hongo, Bunkyo-ku, Tokyo, Japan. rado@m.u-tokyo.ac.jp., Sexton PM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia. patrick.sexton@monash.edu.; School of Pharmacy, Fudan University, Shanghai, China. patrick.sexton@monash.edu., Wootten D; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia. denise.wootten@monash.edu.; School of Pharmacy, Fudan University, Shanghai, China. denise.wootten@monash.edu.
Source: Nature [Nature] 2020 Jan; Vol. 577 (7790), pp. 432-436. Date of Electronic Publication: 2020 Jan 08.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 0410462 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1476-4687 (Electronic) Linking ISSN: 00280836 NLM ISO Abbreviation: Nature Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="AU" term="%22Zhao+P%22">Zhao P</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Liang+YL%22">Liang YL</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Belousoff+MJ%22">Belousoff MJ</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Deganutti+G%22">Deganutti G</searchLink>; School of Biological Sciences, University of Essex, Colchester, UK.<br /><searchLink fieldCode="AU" term="%22Fletcher+MM%22">Fletcher MM</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Willard+FS%22">Willard FS</searchLink>; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA.<br /><searchLink fieldCode="AU" term="%22Bell+MG%22">Bell MG</searchLink>; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA.<br /><searchLink fieldCode="AU" term="%22Christe+ME%22">Christe ME</searchLink>; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA.<br /><searchLink fieldCode="AU" term="%22Sloop+KW%22">Sloop KW</searchLink>; Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, IN, USA.<br /><searchLink fieldCode="AU" term="%22Inoue+A%22">Inoue A</searchLink>; Graduate School of Pharmaceutical Sciences, Tohoku University, Sendai, Miyagi, Japan.<br /><searchLink fieldCode="AU" term="%22Truong+TT%22">Truong TT</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Clydesdale+L%22">Clydesdale L</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Furness+SGB%22">Furness SGB</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Christopoulos+A%22">Christopoulos A</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.<br /><searchLink fieldCode="AU" term="%22Wang+MW%22">Wang MW</searchLink>; The National Center for Drug Screening and CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, China.; School of Pharmacy, Fudan University, Shanghai, China.<br /><searchLink fieldCode="AU" term="%22Miller+LJ%22">Miller LJ</searchLink>; Mayo Clinic, Scottsdale, AZ, USA.<br /><searchLink fieldCode="AU" term="%22Reynolds+CA%22">Reynolds CA</searchLink>; School of Biological Sciences, University of Essex, Colchester, UK.<br /><searchLink fieldCode="AU" term="%22Danev+R%22">Danev R</searchLink>; Graduate School of Medicine, University of Tokyo, Hongo, Bunkyo-ku, Tokyo, Japan. rado@m.u-tokyo.ac.jp.<br /><searchLink fieldCode="AU" term="%22Sexton+PM%22">Sexton PM</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia. patrick.sexton@monash.edu.; School of Pharmacy, Fudan University, Shanghai, China. patrick.sexton@monash.edu.<br /><searchLink fieldCode="AU" term="%22Wootten+D%22">Wootten D</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia. denise.wootten@monash.edu.; School of Pharmacy, Fudan University, Shanghai, China. denise.wootten@monash.edu.
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