Discovery of T-1101 tosylate as a first-in-class clinical candidate for Hec1/Nek2 inhibition in cancer therapy.

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Title: Discovery of T-1101 tosylate as a first-in-class clinical candidate for Hec1/Nek2 inhibition in cancer therapy.
Authors: Chuang SH; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Lee YE; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Huang LYL; Taivex Therapeutics Corporation, 2nd Floor, Dongxing Rd., Songshan Dist., Taipei City, 10511, Taiwan., Chen CK; Genomics Research Center, Academia Sinica, Taipei City, Taiwan., Lai CL; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Lin YH; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Yang JY; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Yang SC; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Chang LH; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Chen CH; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Liu CW; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Lin HS; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Lee YR; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Huang KP; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Fu KC; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Jen HM; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Lai JY; Department of Applied Chemistry, National Chiayi University, No. 300, Syuefu Rd., Chiayi City, 60004, Taiwan., Jian PS; Department of Applied Chemistry, National Chiayi University, No. 300, Syuefu Rd., Chiayi City, 60004, Taiwan., Wang YC; Department of Applied Chemistry, National Chiayi University, No. 300, Syuefu Rd., Chiayi City, 60004, Taiwan., Hsueh WY; Department of Applied Chemistry, National Chiayi University, No. 300, Syuefu Rd., Chiayi City, 60004, Taiwan., Tsai PY; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Hong WH; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Chang CC; Taivex Therapeutics Corporation, 2nd Floor, Dongxing Rd., Songshan Dist., Taipei City, 10511, Taiwan., Wu DZ; Xenobiotic Laboratories, Inc., Plainsboro, NJ, USA., Wu J; Xenobiotic Laboratories, Inc., Plainsboro, NJ, USA., Chen MH; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Yu KM; Taivex Therapeutics Corporation, 2nd Floor, Dongxing Rd., Songshan Dist., Taipei City, 10511, Taiwan., Chern CY; Department of Applied Chemistry, National Chiayi University, No. 300, Syuefu Rd., Chiayi City, 60004, Taiwan., Chang JM; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan., Lau JYN; Taivex Therapeutics Corporation, 2nd Floor, Dongxing Rd., Songshan Dist., Taipei City, 10511, Taiwan., Huang JJ; Development Center for Biotechnology, National Biotechnology Research Park, Taipei City, 11571, Taiwan; Department of Applied Chemistry, National Chiayi University, No. 300, Syuefu Rd., Chiayi City, 60004, Taiwan. Electronic address: lukehuang@mail.ncyu.edu.tw.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2020 Apr 01; Vol. 191, pp. 112118. Date of Electronic Publication: 2020 Feb 07.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1768-3254
DOI:10.1016/j.ejmech.2020.112118