Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation.
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| Title: | Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation. |
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| Authors: | Venugopala KN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Biotechnology and Food Technology, Durban University of Technology, Durban 4001, South Africa., Ramachandra P; Department of Chemistry, School of Applied Sciences, REVA University, Bangalore 560 064, India., Tratrat C; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Gleiser RM; CREAN-IMBIV (UNC-CONICET), Av. Valparaíso s.n., Córdoba, Argentina and FCEFyN, AV. Sarsfield 299, Universidad Nacional de Cordoba, Cordoba 5000, Argentina., Bhandary S; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal By-pass Road, Bhauri, Bhopal 462 066, Madhya Pradesh, India., Chopra D; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal By-pass Road, Bhauri, Bhopal 462 066, Madhya Pradesh, India., Morsy MA; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacology, Faculty of Medicine, Minia University, El-Minia 61511, Egypt., Aldhubiab BE; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Attimarad M; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Nair AB; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Sreeharsha N; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Venugopala R; Department of Public Health Medicine, University of KwaZulu-Natal, Howard College Campus, Durban 4001, South Africa., Deb PK; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan., Chandrashekharappa S; Institute for Stem Cell Biology and Regenerative Medicine, NCBS, TIFR, GKVK, Bellary Road, Bangalore 560 065, India., Khalil HE; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacognosy, Faculty of Pharmacy, Minia University, Minia 61519, Egypt., Alwassil OI; Department of Pharmaceutical Sciences, College of Pharmacy, King Saud bin Abdulaziz University for Health Sciences, Riyadh 11481, Saudi Arabia., Abed SN; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan., Bataineh YA; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan., Palenge R; Department of Chemistry, School of Applied Sciences, REVA University, Bangalore 560 064, India., Haroun M; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Pottathil S; Department of Biomedical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Girish MB; Department of Biomedical Sciences, College of Medicine, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Akrawi SH; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Mohanlall V; Department of Biotechnology and Food Technology, Durban University of Technology, Durban 4001, South Africa. |
| Source: | Molecules (Basel, Switzerland) [Molecules] 2020 Mar 13; Vol. 25 (6). Date of Electronic Publication: 2020 Mar 13. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Links: – Type: pdflink Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 32183140 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Venugopala+KN%22">Venugopala KN</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Biotechnology and Food Technology, Durban University of Technology, Durban 4001, South Africa.<br /><searchLink fieldCode="AU" term="%22Ramachandra+P%22">Ramachandra P</searchLink>; Department of Chemistry, School of Applied Sciences, REVA University, Bangalore 560 064, India.<br /><searchLink fieldCode="AU" term="%22Tratrat+C%22">Tratrat C</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Gleiser+RM%22">Gleiser RM</searchLink>; CREAN-IMBIV (UNC-CONICET), Av. Valparaíso s.n., Córdoba, Argentina and FCEFyN, AV. Sarsfield 299, Universidad Nacional de Cordoba, Cordoba 5000, Argentina.<br /><searchLink fieldCode="AU" term="%22Bhandary+S%22">Bhandary S</searchLink>; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal By-pass Road, Bhauri, Bhopal 462 066, Madhya Pradesh, India.<br /><searchLink fieldCode="AU" term="%22Chopra+D%22">Chopra D</searchLink>; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal By-pass Road, Bhauri, Bhopal 462 066, Madhya Pradesh, India.<br /><searchLink fieldCode="AU" term="%22Morsy+MA%22">Morsy MA</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacology, Faculty of Medicine, Minia University, El-Minia 61511, Egypt.<br /><searchLink fieldCode="AU" term="%22Aldhubiab+BE%22">Aldhubiab BE</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Attimarad+M%22">Attimarad M</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Nair+AB%22">Nair AB</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Sreeharsha+N%22">Sreeharsha N</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Venugopala+R%22">Venugopala R</searchLink>; Department of Public Health Medicine, University of KwaZulu-Natal, Howard College Campus, Durban 4001, South Africa.<br /><searchLink fieldCode="AU" term="%22Deb+PK%22">Deb PK</searchLink>; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan.<br /><searchLink fieldCode="AU" term="%22Chandrashekharappa+S%22">Chandrashekharappa S</searchLink>; Institute for Stem Cell Biology and Regenerative Medicine, NCBS, TIFR, GKVK, Bellary Road, Bangalore 560 065, India.<br /><searchLink fieldCode="AU" term="%22Khalil+HE%22">Khalil HE</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.; Department of Pharmacognosy, Faculty of Pharmacy, Minia University, Minia 61519, Egypt.<br /><searchLink fieldCode="AU" term="%22Alwassil+OI%22">Alwassil OI</searchLink>; Department of Pharmaceutical Sciences, College of Pharmacy, King Saud bin Abdulaziz University for Health Sciences, Riyadh 11481, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Abed+SN%22">Abed SN</searchLink>; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan.<br /><searchLink fieldCode="AU" term="%22Bataineh+YA%22">Bataineh YA</searchLink>; Department of Pharmaceutical Sciences, Faculty of Pharmacy, Philadelphia University, P.O. Box 1, Amman 19392, Jordan.<br /><searchLink fieldCode="AU" term="%22Palenge+R%22">Palenge R</searchLink>; Department of Chemistry, School of Applied Sciences, REVA University, Bangalore 560 064, India.<br /><searchLink fieldCode="AU" term="%22Haroun+M%22">Haroun M</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Pottathil+S%22">Pottathil S</searchLink>; Department of Biomedical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Girish+MB%22">Girish MB</searchLink>; Department of Biomedical Sciences, College of Medicine, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Akrawi+SH%22">Akrawi SH</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa 31982, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Mohanlall+V%22">Mohanlall V</searchLink>; Department of Biotechnology and Food Technology, Durban University of Technology, Durban 4001, South Africa. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22100964009%22">Molecules (Basel, Switzerland)</searchLink> [Molecules] 2020 Mar 13; Vol. 25 (6). <i>Date of Electronic Publication: </i>2020 Mar 13. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22MDPI%22">MDPI </searchLink><i>Country of Publication: </i>Switzerland <i>NLM ID: </i>100964009 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1420-3049 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2214203049%22">14203049 </searchLink><i>NLM ISO Abbreviation: </i>Molecules <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=32183140 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.3390/molecules25061316 Languages: – Code: eng Text: English Titles: – TitleFull: Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Venugopala KN – PersonEntity: Name: NameFull: Ramachandra P – PersonEntity: Name: NameFull: Tratrat C – PersonEntity: Name: NameFull: Gleiser RM – PersonEntity: Name: NameFull: Bhandary S – PersonEntity: Name: NameFull: Chopra D – PersonEntity: Name: NameFull: Morsy MA – PersonEntity: Name: NameFull: Aldhubiab BE – PersonEntity: Name: NameFull: Attimarad M – PersonEntity: Name: NameFull: Nair AB – PersonEntity: Name: NameFull: Sreeharsha N – PersonEntity: Name: NameFull: Venugopala R – PersonEntity: Name: NameFull: Deb PK – PersonEntity: Name: NameFull: Chandrashekharappa S – PersonEntity: Name: NameFull: Khalil HE – PersonEntity: Name: NameFull: Alwassil OI – PersonEntity: Name: NameFull: Abed SN – PersonEntity: Name: NameFull: Bataineh YA – PersonEntity: Name: NameFull: Palenge R – PersonEntity: Name: NameFull: Haroun M – PersonEntity: Name: NameFull: Pottathil S – PersonEntity: Name: NameFull: Girish MB – PersonEntity: Name: NameFull: Akrawi SH – PersonEntity: Name: NameFull: Mohanlall V IsPartOfRelationships: – BibEntity: Dates: – D: 13 M: 03 Text: 2020 Mar 13 Type: published Y: 2020 Identifiers: – Type: issn-electronic Value: 1420-3049 Numbering: – Type: volume Value: 25 – Type: issue Value: 6 Titles: – TitleFull: Molecules (Basel, Switzerland) Type: main |
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