Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties.
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| Title: | Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties. |
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| Authors: | Hudson AR; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States. Electronic address: andyrhudson@gmail.com., Santora VJ; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Petroski RE; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Almos TA; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Anderson G; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Barido R; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Basinger J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Bellows CL; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Bookser BC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Broadbent NJ; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Cabebe C; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Chai CK; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Chen M; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Chow S; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Chung M; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Heger L; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Danks AM; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Freestone GC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Gitnick D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Gupta V; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Hoffmaster C; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Kaplan AP; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Kennedy MR; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Lee D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Limberis J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Ly K; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Mak CC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Masatsugu B; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Morse AC; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Na J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Neul D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Nikpur J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Renick J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Sebring K; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Sevidal S; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Tabatabaei A; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Wen J; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Xia S; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Yan Y; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Yoder ZW; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Zook D; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Peters M; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States., Breitenbucher JG; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States. |
| Source: | Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2020 Jul 15; Vol. 30 (14), pp. 127214. Date of Electronic Publication: 2020 Apr 25. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 32527538 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Hudson+AR%22">Hudson AR</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States. Electronic address: andyrhudson@gmail.com.<br /><searchLink fieldCode="AU" term="%22Santora+VJ%22">Santora VJ</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Petroski+RE%22">Petroski RE</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Almos+TA%22">Almos TA</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Anderson+G%22">Anderson G</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Barido+R%22">Barido R</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Basinger+J%22">Basinger J</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Bellows+CL%22">Bellows CL</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Bookser+BC%22">Bookser BC</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Broadbent+NJ%22">Broadbent NJ</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Cabebe+C%22">Cabebe C</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Chai+CK%22">Chai CK</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Chen+M%22">Chen M</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Chow+S%22">Chow S</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Chung+M%22">Chung M</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Heger+L%22">Heger L</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Danks+AM%22">Danks AM</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Freestone+GC%22">Freestone GC</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Gitnick+D%22">Gitnick D</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Gupta+V%22">Gupta V</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Hoffmaster+C%22">Hoffmaster C</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Kaplan+AP%22">Kaplan AP</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Kennedy+MR%22">Kennedy MR</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Lee+D%22">Lee D</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Limberis+J%22">Limberis J</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Ly+K%22">Ly K</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Mak+CC%22">Mak CC</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Masatsugu+B%22">Masatsugu B</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Morse+AC%22">Morse AC</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Na+J%22">Na J</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Neul+D%22">Neul D</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Nikpur+J%22">Nikpur J</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Renick+J%22">Renick J</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Sebring+K%22">Sebring K</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Sevidal+S%22">Sevidal S</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Tabatabaei+A%22">Tabatabaei A</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Wen+J%22">Wen J</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Xia+S%22">Xia S</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Yan+Y%22">Yan Y</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Yoder+ZW%22">Yoder ZW</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Zook+D%22">Zook D</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Peters+M%22">Peters M</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States.<br /><searchLink fieldCode="AU" term="%22Breitenbucher+JG%22">Breitenbucher JG</searchLink>; Dart Neuroscience, 12278 Scripps Summit Dr, San Diego, CA 92131, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%229107377%22">Bioorganic & medicinal chemistry letters</searchLink> [Bioorg Med Chem Lett] 2020 Jul 15; Vol. 30 (14), pp. 127214. <i>Date of Electronic Publication: </i>2020 Apr 25. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science+Ltd%22">Elsevier Science Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>9107377 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1464-3405 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%220960894X%22">0960894X </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Med Chem Lett <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=32527538 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bmcl.2020.127214 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 127214 Titles: – TitleFull: Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Hudson AR – PersonEntity: Name: NameFull: Santora VJ – PersonEntity: Name: NameFull: Petroski RE – PersonEntity: Name: NameFull: Almos TA – PersonEntity: Name: NameFull: Anderson G – PersonEntity: Name: NameFull: Barido R – PersonEntity: Name: NameFull: Basinger J – PersonEntity: Name: NameFull: Bellows CL – PersonEntity: Name: NameFull: Bookser BC – PersonEntity: Name: NameFull: Broadbent NJ – PersonEntity: Name: NameFull: Cabebe C – PersonEntity: Name: NameFull: Chai CK – PersonEntity: Name: NameFull: Chen M – PersonEntity: Name: NameFull: Chow S – PersonEntity: Name: NameFull: Chung M – PersonEntity: Name: NameFull: Heger L – PersonEntity: Name: NameFull: Danks AM – PersonEntity: Name: NameFull: Freestone GC – PersonEntity: Name: NameFull: Gitnick D – PersonEntity: Name: NameFull: Gupta V – PersonEntity: Name: NameFull: Hoffmaster C – PersonEntity: Name: NameFull: Kaplan AP – PersonEntity: Name: NameFull: Kennedy MR – PersonEntity: Name: NameFull: Lee D – PersonEntity: Name: NameFull: Limberis J – PersonEntity: Name: NameFull: Ly K – PersonEntity: Name: NameFull: Mak CC – PersonEntity: Name: NameFull: Masatsugu B – PersonEntity: Name: NameFull: Morse AC – PersonEntity: Name: NameFull: Na J – PersonEntity: Name: NameFull: Neul D – PersonEntity: Name: NameFull: Nikpur J – PersonEntity: Name: NameFull: Renick J – PersonEntity: Name: NameFull: Sebring K – PersonEntity: Name: NameFull: Sevidal S – PersonEntity: Name: NameFull: Tabatabaei A – PersonEntity: Name: NameFull: Wen J – PersonEntity: Name: NameFull: Xia S – PersonEntity: Name: NameFull: Yan Y – PersonEntity: Name: NameFull: Yoder ZW – PersonEntity: Name: NameFull: Zook D – PersonEntity: Name: NameFull: Peters M – PersonEntity: Name: NameFull: Breitenbucher JG IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 07 Text: 2020 Jul 15 Type: published Y: 2020 Identifiers: – Type: issn-electronic Value: 1464-3405 Numbering: – Type: volume Value: 30 – Type: issue Value: 14 Titles: – TitleFull: Bioorganic & medicinal chemistry letters Type: main |
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