Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase δ.

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Title: Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase δ.
Authors: Spencer JA; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.; Department of Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G1 1XL, United Kingdom., Baldwin IR; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Barton N; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Chung CW; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Convery MA; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Edwards CD; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Jamieson C; Department of Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G1 1XL, United Kingdom., Mallett DN; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Rowedder JE; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Rowland P; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Thomas DA; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom., Hardy CJ; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2020 Jun 03; Vol. 11 (7), pp. 1386-1391. Date of Electronic Publication: 2020 Jun 03 (Print Publication: 2020).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Design and Development of a Macrocyclic Series Targeting Phosphoinositide 3-Kinase δ.
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  Data: <searchLink fieldCode="AU" term="%22Spencer+JA%22">Spencer JA</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.; Department of Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G1 1XL, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Baldwin+IR%22">Baldwin IR</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Barton+N%22">Barton N</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Chung+CW%22">Chung CW</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Convery+MA%22">Convery MA</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Edwards+CD%22">Edwards CD</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Jamieson+C%22">Jamieson C</searchLink>; Department of Pure and Applied Chemistry, University of Strathclyde, 295 Cathedral Street, Glasgow G1 1XL, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Mallett+DN%22">Mallett DN</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Rowedder+JE%22">Rowedder JE</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Rowland+P%22">Rowland P</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Thomas+DA%22">Thomas DA</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.<br /><searchLink fieldCode="AU" term="%22Hardy+CJ%22">Hardy CJ</searchLink>; GSK Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom.
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  Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2020 Jun 03; Vol. 11 (7), pp. 1386-1391. <i>Date of Electronic Publication: </i>2020 Jun 03 (<i>Print Publication: </i>2020).
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE
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        Value: 10.1021/acsmedchemlett.0c00061
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              Text: 2020 Jun 03
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