Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists.
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| Title: | Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists. |
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| Authors: | Shahien M; Chemistry Department, Faculty of Science, Benha University, Benha 13518, Egypt., Elagawany M; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Damanhour University, Damanhour, Egypt., Sitaula S; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Goher SS; Chemistry Department, Faculty of Science, Benha University, Benha 13518, Egypt., Burris SL; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Sanders R; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Avdagic A; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Billon C; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Hegazy L; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Burris TP; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA., Elgendy B; Chemistry Department, Faculty of Science, Benha University, Benha 13518, Egypt; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA. |
| Source: | Bioorganic chemistry [Bioorg Chem] 2020 Sep; Vol. 102, pp. 104079. Date of Electronic Publication: 2020 Jul 07. |
| Publication Type: | Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 32683181 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Shahien+M%22">Shahien M</searchLink>; Chemistry Department, Faculty of Science, Benha University, Benha 13518, Egypt.<br /><searchLink fieldCode="AU" term="%22Elagawany+M%22">Elagawany M</searchLink>; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Damanhour University, Damanhour, Egypt.<br /><searchLink fieldCode="AU" term="%22Sitaula+S%22">Sitaula S</searchLink>; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Goher+SS%22">Goher SS</searchLink>; Chemistry Department, Faculty of Science, Benha University, Benha 13518, Egypt.<br /><searchLink fieldCode="AU" term="%22Burris+SL%22">Burris SL</searchLink>; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Sanders+R%22">Sanders R</searchLink>; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Avdagic+A%22">Avdagic A</searchLink>; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Billon+C%22">Billon C</searchLink>; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Hegazy+L%22">Hegazy L</searchLink>; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Burris+TP%22">Burris TP</searchLink>; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA.<br /><searchLink fieldCode="AU" term="%22Elgendy+B%22">Elgendy B</searchLink>; Chemistry Department, Faculty of Science, Benha University, Benha 13518, Egypt; Department of Pharmaceutical and Administrative Sciences, St. Louis College of Pharmacy, St. Louis, MO 63110, USA; Center for Clinical Pharmacology, Washington University School of Medicine and St. Louis College of Pharmacy, St. Louis, MO 63110, USA. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%221303703%22">Bioorganic chemistry</searchLink> [Bioorg Chem] 2020 Sep; Vol. 102, pp. 104079. <i>Date of Electronic Publication: </i>2020 Jul 07. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>1303703 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1090-2120 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200452068%22">00452068 </searchLink><i>NLM ISO Abbreviation: </i>Bioorg Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=32683181 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.bioorg.2020.104079 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 104079 Titles: – TitleFull: Modulation of estrogen-related receptors subtype selectivity: Conversion of an ERRβ/γ selective agonist to ERRα/β/γ pan agonists. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Shahien M – PersonEntity: Name: NameFull: Elagawany M – PersonEntity: Name: NameFull: Sitaula S – PersonEntity: Name: NameFull: Goher SS – PersonEntity: Name: NameFull: Burris SL – PersonEntity: Name: NameFull: Sanders R – PersonEntity: Name: NameFull: Avdagic A – PersonEntity: Name: NameFull: Billon C – PersonEntity: Name: NameFull: Hegazy L – PersonEntity: Name: NameFull: Burris TP – PersonEntity: Name: NameFull: Elgendy B IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 09 Text: 2020 Sep Type: published Y: 2020 Identifiers: – Type: issn-electronic Value: 1090-2120 Numbering: – Type: volume Value: 102 Titles: – TitleFull: Bioorganic chemistry Type: main |
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