Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate Prodrug.

Saved in:
Bibliographic Details
Title: Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate Prodrug.
Authors: Kung PP, Fan C, Gukasyan HJ, Huang B, Kephart S, Kraus M, Lee JH, Sutton SC, Yamazaki S, Zehnder L
Source: Journal of medicinal chemistry [J Med Chem] 2021 Feb 11; Vol. 64 (3), pp. 1725-1732. Date of Electronic Publication: 2021 Feb 02.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 33529029
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate Prodrug.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22Kung+PP%22">Kung PP</searchLink><br /><searchLink fieldCode="AU" term="%22Fan+C%22">Fan C</searchLink><br /><searchLink fieldCode="AU" term="%22Gukasyan+HJ%22">Gukasyan HJ</searchLink><br /><searchLink fieldCode="AU" term="%22Huang+B%22">Huang B</searchLink><br /><searchLink fieldCode="AU" term="%22Kephart+S%22">Kephart S</searchLink><br /><searchLink fieldCode="AU" term="%22Kraus+M%22">Kraus M</searchLink><br /><searchLink fieldCode="AU" term="%22Lee+JH%22">Lee JH</searchLink><br /><searchLink fieldCode="AU" term="%22Sutton+SC%22">Sutton SC</searchLink><br /><searchLink fieldCode="AU" term="%22Yamazaki+S%22">Yamazaki S</searchLink><br /><searchLink fieldCode="AU" term="%22Zehnder+L%22">Zehnder L</searchLink>
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2021 Feb 11; Vol. 64 (3), pp. 1725-1732. <i>Date of Electronic Publication: </i>2021 Feb 02.
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=33529029
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.1021/acs.jmedchem.0c02112
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 1725
    Titles:
      – TitleFull: Design and Characterization of a Pyridone-Containing EZH2 Inhibitor Phosphate Prodrug.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: Kung PP
      – PersonEntity:
          Name:
            NameFull: Fan C
      – PersonEntity:
          Name:
            NameFull: Gukasyan HJ
      – PersonEntity:
          Name:
            NameFull: Huang B
      – PersonEntity:
          Name:
            NameFull: Kephart S
      – PersonEntity:
          Name:
            NameFull: Kraus M
      – PersonEntity:
          Name:
            NameFull: Lee JH
      – PersonEntity:
          Name:
            NameFull: Sutton SC
      – PersonEntity:
          Name:
            NameFull: Yamazaki S
      – PersonEntity:
          Name:
            NameFull: Zehnder L
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 11
              M: 02
              Text: 2021 Feb 11
              Type: published
              Y: 2021
          Identifiers:
            – Type: issn-electronic
              Value: 1520-4804
          Numbering:
            – Type: volume
              Value: 64
            – Type: issue
              Value: 3
          Titles:
            – TitleFull: Journal of medicinal chemistry
              Type: main
ResultId 1