View in EDS

Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening.

Saved in:
Bibliographic Details
Title: Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening.
Authors: de Heuvel E; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Kooistra AJ; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Edink E; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., van Klaveren S; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Stuijt J; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., van der Meer T; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Sadek P; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Mabille D; Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp, Wilrijk, Belgium., Caljon G; Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp, Wilrijk, Belgium., Maes L; Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp, Wilrijk, Belgium., Siderius M; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., de Esch IJP; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Sterk GJ; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands., Leurs R; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.
Source: Frontiers in chemistry [Front Chem] 2021 Jan 21; Vol. 8, pp. 608030. Date of Electronic Publication: 2021 Jan 21 (Print Publication: 2020).
Publication Type: Journal Article
Journal Info: Publisher: Frontiers Media S.A Country of Publication: Switzerland NLM ID: 101627988 Publication Model: eCollection Cited Medium: Print ISSN: 2296-2646 (Print) Linking ISSN: 22962646 NLM ISO Abbreviation: Front Chem Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
FullText Text:
  Availability: 0
Header DbId: mdl
DbLabel: MEDLINE Ultimate
An: 33553105
AccessLevel: 2
PubType: Academic Journal
PubTypeId: academicJournal
PreciseRelevancyScore: 0
IllustrationInfo
Items – Name: Title
  Label: Title
  Group: Ti
  Data: Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening.
– Name: Author
  Label: Authors
  Group: Au
  Data: <searchLink fieldCode="AU" term="%22de+Heuvel+E%22">de Heuvel E</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Kooistra+AJ%22">Kooistra AJ</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Edink+E%22">Edink E</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22van+Klaveren+S%22">van Klaveren S</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Stuijt+J%22">Stuijt J</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22van+der+Meer+T%22">van der Meer T</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Sadek+P%22">Sadek P</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Mabille+D%22">Mabille D</searchLink>; Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp, Wilrijk, Belgium.<br /><searchLink fieldCode="AU" term="%22Caljon+G%22">Caljon G</searchLink>; Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp, Wilrijk, Belgium.<br /><searchLink fieldCode="AU" term="%22Maes+L%22">Maes L</searchLink>; Laboratory of Microbiology, Parasitology and Hygiene, University of Antwerp, Wilrijk, Belgium.<br /><searchLink fieldCode="AU" term="%22Siderius+M%22">Siderius M</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22de+Esch+IJP%22">de Esch IJP</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Sterk+GJ%22">Sterk GJ</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.<br /><searchLink fieldCode="AU" term="%22Leurs+R%22">Leurs R</searchLink>; Division of Medicinal Chemistry, Amsterdam Institute of Molecular and Life Sciences, Vrije Universiteit Amsterdam, Amsterdam, Netherlands.
– Name: TitleSource
  Label: Source
  Group: Src
  Data: <searchLink fieldCode="JN" term="%22101627988%22">Frontiers in chemistry</searchLink> [Front Chem] 2021 Jan 21; Vol. 8, pp. 608030. <i>Date of Electronic Publication: </i>2021 Jan 21 (<i>Print Publication: </i>2020).
– Name: TypePub
  Label: Publication Type
  Group: TypPub
  Data: Journal Article
– Name: TitleSource
  Label: Journal Info
  Group: Src
  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Frontiers+Media+S%2EA%22">Frontiers Media S.A </searchLink><i>Country of Publication: </i>Switzerland <i>NLM ID: </i>101627988 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>2296-2646 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2222962646%22">22962646 </searchLink><i>NLM ISO Abbreviation: </i>Front Chem <i>Subsets: </i>PubMed not MEDLINE
PLink https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=33553105
RecordInfo BibRecord:
  BibEntity:
    Identifiers:
      – Type: doi
        Value: 10.3389/fchem.2020.608030
    Languages:
      – Code: eng
        Text: English
    PhysicalDescription:
      Pagination:
        StartPage: 608030
    Titles:
      – TitleFull: Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening.
        Type: main
  BibRelationships:
    HasContributorRelationships:
      – PersonEntity:
          Name:
            NameFull: de Heuvel E
      – PersonEntity:
          Name:
            NameFull: Kooistra AJ
      – PersonEntity:
          Name:
            NameFull: Edink E
      – PersonEntity:
          Name:
            NameFull: van Klaveren S
      – PersonEntity:
          Name:
            NameFull: Stuijt J
      – PersonEntity:
          Name:
            NameFull: van der Meer T
      – PersonEntity:
          Name:
            NameFull: Sadek P
      – PersonEntity:
          Name:
            NameFull: Mabille D
      – PersonEntity:
          Name:
            NameFull: Caljon G
      – PersonEntity:
          Name:
            NameFull: Maes L
      – PersonEntity:
          Name:
            NameFull: Siderius M
      – PersonEntity:
          Name:
            NameFull: de Esch IJP
      – PersonEntity:
          Name:
            NameFull: Sterk GJ
      – PersonEntity:
          Name:
            NameFull: Leurs R
    IsPartOfRelationships:
      – BibEntity:
          Dates:
            – D: 21
              M: 01
              Text: 2021 Jan 21
              Type: published
              Y: 2021
          Identifiers:
            – Type: issn-print
              Value: 2296-2646
          Numbering:
            – Type: volume
              Value: 8
          Titles:
            – TitleFull: Frontiers in chemistry
              Type: main
ResultId 1