Phenotypic screen identifies calcineurin-sparing FK506 analogs as BMP potentiators for treatment of acute kidney injury.

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Title: Phenotypic screen identifies calcineurin-sparing FK506 analogs as BMP potentiators for treatment of acute kidney injury.
Authors: Larraufie MH; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Gao X; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Xia X; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Devine PJ; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Kallen J; Novartis Institutes for Biomedical Research, Basel, Switzerland., Liu D; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Michaud G; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Harsch A; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Savage N; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Ding J; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Tan K; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Mihalic M; Novartis Institutes for Biomedical Research, Basel, Switzerland., Roggo S; Novartis Institutes for Biomedical Research, Basel, Switzerland., Canham SM; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Bushell SM; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Krastel P; Novartis Institutes for Biomedical Research, Basel, Switzerland., Gao J; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Izaac A; Novartis Institutes for Biomedical Research, Basel, Switzerland., Altinoglu E; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Lustenberger P; Novartis Global Drug Development, Basel, Switzerland., Salcius M; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Harbinski F; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Williams ET; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Zeng L; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Loureiro J; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Cong F; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Fryer CJ; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Klickstein L; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Tallarico JA; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Jain RK; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Rothman DM; Novartis Institutes for Biomedical Research, Cambridge, MA, USA., Wang S; Novartis Institutes for Biomedical Research, Cambridge, MA, USA. Electronic address: shaowen.wang@novartis.com.
Source: Cell chemical biology [Cell Chem Biol] 2021 Sep 16; Vol. 28 (9), pp. 1271-1282.e12. Date of Electronic Publication: 2021 Apr 23.
Publication Type: Journal Article
Journal Info: Publisher: Cell Press Country of Publication: United States NLM ID: 101676030 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2451-9448 (Electronic) Linking ISSN: 24519448 NLM ISO Abbreviation: Cell Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:2451-9448
DOI:10.1016/j.chembiol.2021.04.001