Single- and Multiple-Dose Pharmacokinetics and Pharmacodynamics of PN-943, a Gastrointestinal-Restricted Oral Peptide Antagonist of α4β7, in Healthy Volunteers.

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Title: Single- and Multiple-Dose Pharmacokinetics and Pharmacodynamics of PN-943, a Gastrointestinal-Restricted Oral Peptide Antagonist of α4β7, in Healthy Volunteers.
Authors: Modi NB; Protagonist Therapeutics, Inc, Newark, California, USA., Cheng X; Protagonist Therapeutics, Inc, Newark, California, USA., Mattheakis L; Protagonist Therapeutics, Inc, Newark, California, USA., Hwang CC; Protagonist Therapeutics, Inc, Newark, California, USA., Nawabi R; Protagonist Therapeutics, Inc, Newark, California, USA., Liu D; Protagonist Therapeutics, Inc, Newark, California, USA., Gupta S; Protagonist Therapeutics, Inc, Newark, California, USA.
Source: Clinical pharmacology in drug development [Clin Pharmacol Drug Dev] 2021 Nov; Vol. 10 (11), pp. 1263-1278. Date of Electronic Publication: 2021 May 04.
Publication Type: Journal Article; Randomized Controlled Trial; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Wiley Country of Publication: United States NLM ID: 101572899 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 2160-7648 (Electronic) Linking ISSN: 2160763X NLM ISO Abbreviation: Clin Pharmacol Drug Dev Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:2160-7648
DOI:10.1002/cpdd.946