Anti-tubercular activity and molecular docking studies of indolizine derivatives targeting mycobacterial InhA enzyme.

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Title: Anti-tubercular activity and molecular docking studies of indolizine derivatives targeting mycobacterial InhA enzyme.
Authors: Venugopala KN; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Department of Biotechnology and Food Technology, Durban University of Technology, Durban, South Africa., Chandrashekharappa S; Institute for Stem Cell Science and Regenerative Medicine (inStem), Bangalore, India., Deb PK; Faculty of Pharmacy, Department of Pharmaceutical Sciences, Philadelphia University, Amman, Jordan., Tratrat C; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia., Pillay M; Department of Microbiology, National Health Laboratory Services, KZN Academic Complex, Inkosi Albert Luthuli Central Hospital, Durban, South Africa., Chopra D; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal, India., Al-Shar'i NA; Faculty of Pharmacy, Department of Medicinal Chemistry and Pharmacognosy, Jordan University of Science and Technology, Irbid, Jordan., Hourani W; Faculty of Pharmacy, Department of Pharmaceutical Sciences, Philadelphia University, Amman, Jordan., Dahabiyeh LA; Department of Pharmaceutical Sciences, School of Pharmacy, The University of Jordan, Amman, Jordan., Borah P; Pratiksha Institute of Pharmaceutical Sciences, Guwahati, India., Nagdeve RD; Department of Chemistry, Visvesvaraya National Institute of Technology, Nagpur, India., Nayak SK; Department of Chemistry, Visvesvaraya National Institute of Technology, Nagpur, India., Padmashali B; Department of Chemistry, School of Basic Science, Rani Channamma University, Belagavi, India., Morsy MA; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Faculty of Medicine, Department of Pharmacology, Minia University, El-Minia, Egypt., Aldhubiab BE; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia., Attimarad M; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia., Nair AB; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia., Sreeharsha N; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Department of Pharmaceutics, Vidya Siri College of Pharmacy, Bangalore, India., Haroun M; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia., Shashikanth S; Department of Studies in Organic Chemistry, University of Mysore, Mysore, India., Mohanlall V; Department of Biotechnology and Food Technology, Durban University of Technology, Durban, South Africa., Mailavaram R; Pharmaceutical Chemistry Division, Sri Vishnu College of Pharmacy, Bhimavaram, India.
Source: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2021 Dec; Vol. 36 (1), pp. 1472-1487.
Publication Type: Journal Article
Journal Info: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Anti-tubercular activity and molecular docking studies of indolizine derivatives targeting mycobacterial InhA enzyme.
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  Data: <searchLink fieldCode="AU" term="%22Venugopala+KN%22">Venugopala KN</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Department of Biotechnology and Food Technology, Durban University of Technology, Durban, South Africa.<br /><searchLink fieldCode="AU" term="%22Chandrashekharappa+S%22">Chandrashekharappa S</searchLink>; Institute for Stem Cell Science and Regenerative Medicine (inStem), Bangalore, India.<br /><searchLink fieldCode="AU" term="%22Deb+PK%22">Deb PK</searchLink>; Faculty of Pharmacy, Department of Pharmaceutical Sciences, Philadelphia University, Amman, Jordan.<br /><searchLink fieldCode="AU" term="%22Tratrat+C%22">Tratrat C</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Pillay+M%22">Pillay M</searchLink>; Department of Microbiology, National Health Laboratory Services, KZN Academic Complex, Inkosi Albert Luthuli Central Hospital, Durban, South Africa.<br /><searchLink fieldCode="AU" term="%22Chopra+D%22">Chopra D</searchLink>; Department of Chemistry, Indian Institute of Science Education and Research Bhopal, Bhopal, India.<br /><searchLink fieldCode="AU" term="%22Al-Shar'i+NA%22">Al-Shar'i NA</searchLink>; Faculty of Pharmacy, Department of Medicinal Chemistry and Pharmacognosy, Jordan University of Science and Technology, Irbid, Jordan.<br /><searchLink fieldCode="AU" term="%22Hourani+W%22">Hourani W</searchLink>; Faculty of Pharmacy, Department of Pharmaceutical Sciences, Philadelphia University, Amman, Jordan.<br /><searchLink fieldCode="AU" term="%22Dahabiyeh+LA%22">Dahabiyeh LA</searchLink>; Department of Pharmaceutical Sciences, School of Pharmacy, The University of Jordan, Amman, Jordan.<br /><searchLink fieldCode="AU" term="%22Borah+P%22">Borah P</searchLink>; Pratiksha Institute of Pharmaceutical Sciences, Guwahati, India.<br /><searchLink fieldCode="AU" term="%22Nagdeve+RD%22">Nagdeve RD</searchLink>; Department of Chemistry, Visvesvaraya National Institute of Technology, Nagpur, India.<br /><searchLink fieldCode="AU" term="%22Nayak+SK%22">Nayak SK</searchLink>; Department of Chemistry, Visvesvaraya National Institute of Technology, Nagpur, India.<br /><searchLink fieldCode="AU" term="%22Padmashali+B%22">Padmashali B</searchLink>; Department of Chemistry, School of Basic Science, Rani Channamma University, Belagavi, India.<br /><searchLink fieldCode="AU" term="%22Morsy+MA%22">Morsy MA</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Faculty of Medicine, Department of Pharmacology, Minia University, El-Minia, Egypt.<br /><searchLink fieldCode="AU" term="%22Aldhubiab+BE%22">Aldhubiab BE</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Attimarad+M%22">Attimarad M</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Nair+AB%22">Nair AB</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Sreeharsha+N%22">Sreeharsha N</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.; Department of Pharmaceutics, Vidya Siri College of Pharmacy, Bangalore, India.<br /><searchLink fieldCode="AU" term="%22Haroun+M%22">Haroun M</searchLink>; Department of Pharmaceutical Sciences, College of Clinical Pharmacy, King Faisal University, Al-Ahsa, Saudi Arabia.<br /><searchLink fieldCode="AU" term="%22Shashikanth+S%22">Shashikanth S</searchLink>; Department of Studies in Organic Chemistry, University of Mysore, Mysore, India.<br /><searchLink fieldCode="AU" term="%22Mohanlall+V%22">Mohanlall V</searchLink>; Department of Biotechnology and Food Technology, Durban University of Technology, Durban, South Africa.<br /><searchLink fieldCode="AU" term="%22Mailavaram+R%22">Mailavaram R</searchLink>; Pharmaceutical Chemistry Division, Sri Vishnu College of Pharmacy, Bhimavaram, India.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Taylor+%26+Francis%22">Taylor & Francis </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101150203 <i>Publication Model: </i>Print <i>Cited Medium: </i>Internet <i>ISSN: </i>1475-6374 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2214756366%22">14756366 </searchLink><i>NLM ISO Abbreviation: </i>J Enzyme Inhib Med Chem <i>Subsets: </i>MEDLINE
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