Rapid Evaluation of Small Molecule Cellular Target Engagement with a Luminescent Thermal Shift Assay.

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Title: Rapid Evaluation of Small Molecule Cellular Target Engagement with a Luminescent Thermal Shift Assay.
Authors: Mortison JD; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States., Cornella-Taracido I; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States., Venkatchalam G; Quantitative Biosciences, MSD, Singapore 138665, Singapore., Partridge AW; Quantitative Biosciences, MSD, Singapore 138665, Singapore., Siriwardana N; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States., Bushell SM; Chemical Biology, Merck & Co., Inc., Boston, Massachusetts 02115, United States.
Source: ACS medicinal chemistry letters [ACS Med Chem Lett] 2021 Jul 12; Vol. 12 (8), pp. 1288-1294. Date of Electronic Publication: 2021 Jul 12 (Print Publication: 2021).
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2021 Jul 12; Vol. 12 (8), pp. 1288-1294. <i>Date of Electronic Publication: </i>2021 Jul 12 (<i>Print Publication: </i>2021).
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE
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        Value: 10.1021/acsmedchemlett.1c00276
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              Text: 2021 Jul 12
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