AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss.
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| Title: | AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss. |
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| Authors: | Hati S; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Zallocchi M; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Hazlitt R; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA., Li Y; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Vijayakumar S; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Min J; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA., Rankovic Z; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA., Lovas S; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Zuo J; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA. Electronic address: jianzuo@creighton.edu. |
| Source: | European journal of medicinal chemistry [Eur J Med Chem] 2021 Dec 15; Vol. 226, pp. 113849. Date of Electronic Publication: 2021 Sep 20. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 34560429 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Hati+S%22">Hati S</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Zallocchi+M%22">Zallocchi M</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Hazlitt+R%22">Hazlitt R</searchLink>; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA.<br /><searchLink fieldCode="AU" term="%22Li+Y%22">Li Y</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Vijayakumar+S%22">Vijayakumar S</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Min+J%22">Min J</searchLink>; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA.<br /><searchLink fieldCode="AU" term="%22Rankovic+Z%22">Rankovic Z</searchLink>; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA.<br /><searchLink fieldCode="AU" term="%22Lovas+S%22">Lovas S</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Zuo+J%22">Zuo J</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA. Electronic address: jianzuo@creighton.edu. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%220420510%22">European journal of medicinal chemistry</searchLink> [Eur J Med Chem] 2021 Dec 15; Vol. 226, pp. 113849. <i>Date of Electronic Publication: </i>2021 Sep 20. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Editions+Scientifiques+Elsevier%22">Editions Scientifiques Elsevier </searchLink><i>Country of Publication: </i>France <i>NLM ID: </i>0420510 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1768-3254 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2202235234%22">02235234 </searchLink><i>NLM ISO Abbreviation: </i>Eur J Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=34560429 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.ejmech.2021.113849 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 113849 Titles: – TitleFull: AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Hati S – PersonEntity: Name: NameFull: Zallocchi M – PersonEntity: Name: NameFull: Hazlitt R – PersonEntity: Name: NameFull: Li Y – PersonEntity: Name: NameFull: Vijayakumar S – PersonEntity: Name: NameFull: Min J – PersonEntity: Name: NameFull: Rankovic Z – PersonEntity: Name: NameFull: Lovas S – PersonEntity: Name: NameFull: Zuo J IsPartOfRelationships: – BibEntity: Dates: – D: 15 M: 12 Text: 2021 Dec 15 Type: published Y: 2021 Identifiers: – Type: issn-electronic Value: 1768-3254 Numbering: – Type: volume Value: 226 Titles: – TitleFull: European journal of medicinal chemistry Type: main |
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