AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss.

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Title: AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss.
Authors: Hati S; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Zallocchi M; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Hazlitt R; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA., Li Y; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Vijayakumar S; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Min J; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA., Rankovic Z; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA., Lovas S; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA., Zuo J; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA. Electronic address: jianzuo@creighton.edu.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2021 Dec 15; Vol. 226, pp. 113849. Date of Electronic Publication: 2021 Sep 20.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: AZD5438-PROTAC: A selective CDK2 degrader that protects against cisplatin- and noise-induced hearing loss.
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  Data: <searchLink fieldCode="AU" term="%22Hati+S%22">Hati S</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Zallocchi+M%22">Zallocchi M</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Hazlitt+R%22">Hazlitt R</searchLink>; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA.<br /><searchLink fieldCode="AU" term="%22Li+Y%22">Li Y</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Vijayakumar+S%22">Vijayakumar S</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Min+J%22">Min J</searchLink>; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA.<br /><searchLink fieldCode="AU" term="%22Rankovic+Z%22">Rankovic Z</searchLink>; Department of Chemical Biology & Therapeutics, St. Jude Children's Research Hospital, Memphis, TN, 38105, USA.<br /><searchLink fieldCode="AU" term="%22Lovas+S%22">Lovas S</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA.<br /><searchLink fieldCode="AU" term="%22Zuo+J%22">Zuo J</searchLink>; Department of Biomedical Sciences, School of Medicine, Creighton University, Omaha, NE, 68178, USA. Electronic address: jianzuo@creighton.edu.
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              Text: 2021 Dec 15
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