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PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation.

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Title: PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation.
Authors: Machulkin AE; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation. Electronic address: alekseymachulkin@rambler.ru., Uspenskaya AA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Zyk NY; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Nimenko EA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Ber AP; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Petrov SA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Shafikov RR; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow, 117997, Russian Federation., Skvortsov DA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Faculty of Biology and Biotechnologies, Higher School of Economics, Myasnitskaya 13, Moscow, 101000, Russia., Smirnova GB; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia., Borisova YA; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia., Pokrovsky VS; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia; RUDN University, Miklukho-Maklaya Str.6, Moscow, 117198, Russian Federation., Kolmogorov VS; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Vaneev AN; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Ivanenkov YA; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Moscow Institute of Physics and Technology (State University), 9 Institutskiy Lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russia; Institute of Biochemistry and Genetics Ufa Science Centre Russian Academy of Sciences (IBG RAS), Oktyabrya Prospekt 71, Ufa, 450054, Russian Federation., Khudyakov AD; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Kovalev SV; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Erofeev AS; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Gorelkin PV; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation., Beloglazkina EK; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Zyk NV; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation., Khazanova ES; LLC Izvarino-Pharma, V. Vnukovskoe, Vnukovskoe Sh., 5th Km., Building 1, Moscow, 108817, Russian Federation., Majouga AG; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow, 125047, Russian Federation.
Source: European journal of medicinal chemistry [Eur J Med Chem] 2022 Jan 05; Vol. 227, pp. 113936. Date of Electronic Publication: 2021 Oct 23.
Publication Type: Journal Article
Journal Info: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE
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  Data: PSMA-targeted small-molecule docetaxel conjugate: Synthesis and preclinical evaluation.
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  Data: <searchLink fieldCode="AU" term="%22Machulkin+AE%22">Machulkin AE</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation. Electronic address: alekseymachulkin@rambler.ru.<br /><searchLink fieldCode="AU" term="%22Uspenskaya+AA%22">Uspenskaya AA</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Zyk+NY%22">Zyk NY</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Nimenko+EA%22">Nimenko EA</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Ber+AP%22">Ber AP</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Petrov+SA%22">Petrov SA</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Shafikov+RR%22">Shafikov RR</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Shemyakin and Ovchinnikov Institute of Bioorganic Chemistry Russian Academy of Sciences, GSP-7, Ulitsa Miklukho-Maklaya, 16/10, Moscow, 117997, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Skvortsov+DA%22">Skvortsov DA</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Faculty of Biology and Biotechnologies, Higher School of Economics, Myasnitskaya 13, Moscow, 101000, Russia.<br /><searchLink fieldCode="AU" term="%22Smirnova+GB%22">Smirnova GB</searchLink>; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia.<br /><searchLink fieldCode="AU" term="%22Borisova+YA%22">Borisova YA</searchLink>; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia.<br /><searchLink fieldCode="AU" term="%22Pokrovsky+VS%22">Pokrovsky VS</searchLink>; N.N. Blokhin Cancer Research Center, 24 Kashirskoye Sh., Moscow, 115478, Russia; RUDN University, Miklukho-Maklaya Str.6, Moscow, 117198, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Kolmogorov+VS%22">Kolmogorov VS</searchLink>; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Vaneev+AN%22">Vaneev AN</searchLink>; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Ivanenkov+YA%22">Ivanenkov YA</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; Moscow Institute of Physics and Technology (State University), 9 Institutskiy Lane, Dolgoprudny City, Moscow Region, 141700, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation; The Federal State Unitary Enterprise Dukhov Automatics Research Institute, Moscow, 127055, Russia; Institute of Biochemistry and Genetics Ufa Science Centre Russian Academy of Sciences (IBG RAS), Oktyabrya Prospekt 71, Ufa, 450054, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Khudyakov+AD%22">Khudyakov AD</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Kovalev+SV%22">Kovalev SV</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Erofeev+AS%22">Erofeev AS</searchLink>; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Gorelkin+PV%22">Gorelkin PV</searchLink>; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Beloglazkina+EK%22">Beloglazkina EK</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Zyk+NV%22">Zyk NV</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Khazanova+ES%22">Khazanova ES</searchLink>; LLC Izvarino-Pharma, V. Vnukovskoe, Vnukovskoe Sh., 5th Km., Building 1, Moscow, 108817, Russian Federation.<br /><searchLink fieldCode="AU" term="%22Majouga+AG%22">Majouga AG</searchLink>; Lomonosov Moscow State University, Chemistry Dept., Leninskie Gory, Building 1/3, GSP-1, Moscow, 119991, Russian Federation; National University of Science and Technology MISiS, 9 Leninskiy Pr, Moscow, 119049, Russian Federation; Dmitry Mendeleev University of Chemical Technology of Russia, Miusskaya Sq. 9, Moscow, 125047, Russian Federation.
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  Data: <searchLink fieldCode="JN" term="%220420510%22">European journal of medicinal chemistry</searchLink> [Eur J Med Chem] 2022 Jan 05; Vol. 227, pp. 113936. <i>Date of Electronic Publication: </i>2021 Oct 23.
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