Co-targeting BET bromodomain BRD4 and RAC1 suppresses growth, stemness and tumorigenesis by disrupting the c-MYC-G9a-FTH1axis and downregulating HDAC1 in molecular subtypes of breast cancer.

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Title: Co-targeting BET bromodomain BRD4 and RAC1 suppresses growth, stemness and tumorigenesis by disrupting the c-MYC-G9a-FTH1axis and downregulating HDAC1 in molecular subtypes of breast cancer.
Authors: Ali A; Research Institute of Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates., Shafarin J; Research Institute of Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates., Unnikannan H; Research Institute of Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates., Al-Jabi N; Department of Basic Medical Sciences, College of Medicine, University of Sharjah, Sharjah, United Arab Emirates., Jabal RA; Department of Basic Medical Sciences, College of Medicine, University of Sharjah, Sharjah, United Arab Emirates., Bajbouj K; Research Institute of Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates.; Department of Basic Medical Sciences, College of Medicine, University of Sharjah, Sharjah, United Arab Emirates., Muhammad JS; Research Institute of Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates.; Department of Basic Medical Sciences, College of Medicine, University of Sharjah, Sharjah, United Arab Emirates., Hamad M; Research Institute of Medical and Health Sciences, University of Sharjah, Sharjah, United Arab Emirates.; Department of Medical Laboratory Sciences, College of Health Sciences, University of Sharjah, Sharjah, United Arab Emirates.
Source: International journal of biological sciences [Int J Biol Sci] 2021 Oct 25; Vol. 17 (15), pp. 4474-4492. Date of Electronic Publication: 2021 Oct 25 (Print Publication: 2021).
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Ivyspring International Country of Publication: Australia NLM ID: 101235568 Publication Model: eCollection Cited Medium: Internet ISSN: 1449-2288 (Electronic) Linking ISSN: 14492288 NLM ISO Abbreviation: Int J Biol Sci Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1449-2288
DOI:10.7150/ijbs.62236