Antitarget Selectivity and Tolerability of Novel Pyrrolo[2,3-d]pyrimidine RET Inhibitors.
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| Title: | Antitarget Selectivity and Tolerability of Novel Pyrrolo[2,3-d]pyrimidine RET Inhibitors. |
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| Authors: | Mathison CJN; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Yang Y; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Nelson J; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Huang Z; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Jiang J; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Chianelli D; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Rucker PV; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Roland J; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Xie YF; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Epple R; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Bursulaya B; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Lee C; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Gao MY; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Shaffer J; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Briones S; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Sarkisova Y; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Galkin A; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Li L; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Li N; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Li C; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Hua S; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Kasibhatla S; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Kinyamu-Akunda J; Novartis Institutes for BioMedical Research, One Health Plaza, East Hanover, New Jersey 07936, United States., Kikkawa R; Novartis Institutes for BioMedical Research, One Health Plaza, East Hanover, New Jersey 07936, United States., Molteni V; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States., Tellew JE; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2021 Nov 06; Vol. 12 (12), pp. 1912-1919. Date of Electronic Publication: 2021 Nov 06 (Print Publication: 2021). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 34917254 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Antitarget Selectivity and Tolerability of Novel Pyrrolo[2,3-d]pyrimidine RET Inhibitors. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Mathison+CJN%22">Mathison CJN</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Yang+Y%22">Yang Y</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Nelson+J%22">Nelson J</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Huang+Z%22">Huang Z</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Jiang+J%22">Jiang J</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Chianelli+D%22">Chianelli D</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Rucker+PV%22">Rucker PV</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Roland+J%22">Roland J</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Xie+YF%22">Xie YF</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Epple+R%22">Epple R</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Bursulaya+B%22">Bursulaya B</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Lee+C%22">Lee C</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Gao+MY%22">Gao MY</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Shaffer+J%22">Shaffer J</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Briones+S%22">Briones S</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Sarkisova+Y%22">Sarkisova Y</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Galkin+A%22">Galkin A</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Li+L%22">Li L</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Li+N%22">Li N</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Li+C%22">Li C</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Hua+S%22">Hua S</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Kasibhatla+S%22">Kasibhatla S</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Kinyamu-Akunda+J%22">Kinyamu-Akunda J</searchLink>; Novartis Institutes for BioMedical Research, One Health Plaza, East Hanover, New Jersey 07936, United States.<br /><searchLink fieldCode="AU" term="%22Kikkawa+R%22">Kikkawa R</searchLink>; Novartis Institutes for BioMedical Research, One Health Plaza, East Hanover, New Jersey 07936, United States.<br /><searchLink fieldCode="AU" term="%22Molteni+V%22">Molteni V</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Tellew+JE%22">Tellew JE</searchLink>; The Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2021 Nov 06; Vol. 12 (12), pp. 1912-1919. <i>Date of Electronic Publication: </i>2021 Nov 06 (<i>Print Publication: </i>2021). – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=34917254 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acsmedchemlett.1c00450 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1912 Titles: – TitleFull: Antitarget Selectivity and Tolerability of Novel Pyrrolo[2,3-d]pyrimidine RET Inhibitors. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Mathison CJN – PersonEntity: Name: NameFull: Yang Y – PersonEntity: Name: NameFull: Nelson J – PersonEntity: Name: NameFull: Huang Z – PersonEntity: Name: NameFull: Jiang J – PersonEntity: Name: NameFull: Chianelli D – PersonEntity: Name: NameFull: Rucker PV – PersonEntity: Name: NameFull: Roland J – PersonEntity: Name: NameFull: Xie YF – PersonEntity: Name: NameFull: Epple R – PersonEntity: Name: NameFull: Bursulaya B – PersonEntity: Name: NameFull: Lee C – PersonEntity: Name: NameFull: Gao MY – PersonEntity: Name: NameFull: Shaffer J – PersonEntity: Name: NameFull: Briones S – PersonEntity: Name: NameFull: Sarkisova Y – PersonEntity: Name: NameFull: Galkin A – PersonEntity: Name: NameFull: Li L – PersonEntity: Name: NameFull: Li N – PersonEntity: Name: NameFull: Li C – PersonEntity: Name: NameFull: Hua S – PersonEntity: Name: NameFull: Kasibhatla S – PersonEntity: Name: NameFull: Kinyamu-Akunda J – PersonEntity: Name: NameFull: Kikkawa R – PersonEntity: Name: NameFull: Molteni V – PersonEntity: Name: NameFull: Tellew JE IsPartOfRelationships: – BibEntity: Dates: – D: 06 M: 11 Text: 2021 Nov 06 Type: published Y: 2021 Identifiers: – Type: issn-print Value: 1948-5875 Numbering: – Type: volume Value: 12 – Type: issue Value: 12 Titles: – TitleFull: ACS medicinal chemistry letters Type: main |
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