CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.

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Title: CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.
Authors: Tomassi S; Dipartimento di Farmacia, Università degli Studi di Napoli 'Federico II', Via D. Montesano 49, Naples 80131, Italy., Dimmito MP; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy., Cai M; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., D'Aniello A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Del Bene A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Messere A; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Liu Z; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., Zhu T; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., Hruby VJ; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States., Stefanucci A; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy., Cosconati S; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy., Mollica A; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy., Di Maro S; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.
Source: Journal of medicinal chemistry [J Med Chem] 2022 Mar 10; Vol. 65 (5), pp. 4007-4017. Date of Electronic Publication: 2022 Feb 21.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: <searchLink fieldCode="AU" term="%22Tomassi+S%22">Tomassi S</searchLink>; Dipartimento di Farmacia, Università degli Studi di Napoli 'Federico II', Via D. Montesano 49, Naples 80131, Italy.<br /><searchLink fieldCode="AU" term="%22Dimmito+MP%22">Dimmito MP</searchLink>; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy.<br /><searchLink fieldCode="AU" term="%22Cai+M%22">Cai M</searchLink>; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.<br /><searchLink fieldCode="AU" term="%22D'Aniello+A%22">D'Aniello A</searchLink>; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.<br /><searchLink fieldCode="AU" term="%22Del+Bene+A%22">Del Bene A</searchLink>; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.<br /><searchLink fieldCode="AU" term="%22Messere+A%22">Messere A</searchLink>; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.<br /><searchLink fieldCode="AU" term="%22Liu+Z%22">Liu Z</searchLink>; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.<br /><searchLink fieldCode="AU" term="%22Zhu+T%22">Zhu T</searchLink>; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.<br /><searchLink fieldCode="AU" term="%22Hruby+VJ%22">Hruby VJ</searchLink>; Department of Chemistry and Biochemistry, University of Arizona, Tucson, Arizona 85721, United States.<br /><searchLink fieldCode="AU" term="%22Stefanucci+A%22">Stefanucci A</searchLink>; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy.<br /><searchLink fieldCode="AU" term="%22Cosconati+S%22">Cosconati S</searchLink>; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.<br /><searchLink fieldCode="AU" term="%22Mollica+A%22">Mollica A</searchLink>; Dipartimento di Farmacia, Università di Chieti-Pescara 'G. d'Annunzio', Via dei Vestini 31, Chieti 66100, Italy.<br /><searchLink fieldCode="AU" term="%22Di+Maro+S%22">Di Maro S</searchLink>; DiSTABiF, University of Campania 'Luigi Vanvitelli', Via Vivaldi 43, 81100 Caserta, Italy.
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2022 Mar 10; Vol. 65 (5), pp. 4007-4017. <i>Date of Electronic Publication: </i>2022 Feb 21.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>9716531 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1520-4804 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200222623%22">00222623 </searchLink><i>NLM ISO Abbreviation: </i>J Med Chem <i>Subsets: </i>MEDLINE
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        Value: 10.1021/acs.jmedchem.1c01848
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              Text: 2022 Mar 10
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