Synthesis and Characterization of Transition-State Analogue Inhibitors against Human DNA Methyltransferase 1.
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| Title: | Synthesis and Characterization of Transition-State Analogue Inhibitors against Human DNA Methyltransferase 1. |
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| Authors: | Lamiable-Oulaidi F; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Harijan RK; Biochemistry Department, Albert Einstein College of Medicine, 1300 Morris Park Avenue, Bronx, New York 10461, United States., Shaffer KJ; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Crump DR; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Sun Y; Biochemistry Department, Albert Einstein College of Medicine, 1300 Morris Park Avenue, Bronx, New York 10461, United States., Du Q; Biochemistry Department, Albert Einstein College of Medicine, 1300 Morris Park Avenue, Bronx, New York 10461, United States., Gulab SA; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Khan AA; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Luxenburger A; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Woolhouse AD; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Sidoli S; Biochemistry Department, Albert Einstein College of Medicine, 1300 Morris Park Avenue, Bronx, New York 10461, United States., Tyler PC; The Ferrier Research Institute, Victoria University of Wellington, P.O. Box 33436, Petone 5046, New Zealand., Schramm VL; Biochemistry Department, Albert Einstein College of Medicine, 1300 Morris Park Avenue, Bronx, New York 10461, United States. |
| Source: | Journal of medicinal chemistry [J Med Chem] 2022 Apr 14; Vol. 65 (7), pp. 5462-5494. Date of Electronic Publication: 2022 Mar 24. |
| Publication Type: | Journal Article; Research Support, Non-U.S. Gov't |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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