Lead Optimization to Advance Protease-Activated Receptor-1 Antagonists in Early Discovery.

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Title: Lead Optimization to Advance Protease-Activated Receptor-1 Antagonists in Early Discovery.
Authors: Mandal M, Madeira M, Amin RP, Buevich AV, Cheng A, Labroli M, Liu X, Acton J, Pio B, Basso A, Chobanian H, Dong G, Dropinski J, Guo Y, Guo Z, Kurowski S, Korfmacher W, Lee S, Meng D, Ondeyka D, Yang Z, Zhang R, Wei H, Wu Z, Zhang F, Wollenberg G, Biftu T, Greenlee WJ, Chintala M, Maletic M, Zhu Z
Source: Journal of medicinal chemistry [J Med Chem] 2022 Apr 14; Vol. 65 (7), pp. 5575-5592. Date of Electronic Publication: 2022 Mar 29.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-4804 (Electronic) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE
Database: MEDLINE Ultimate
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DbLabel: MEDLINE Ultimate
An: 35349275
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PubType: Academic Journal
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PreciseRelevancyScore: 0
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  Data: <searchLink fieldCode="JN" term="%229716531%22">Journal of medicinal chemistry</searchLink> [J Med Chem] 2022 Apr 14; Vol. 65 (7), pp. 5575-5592. <i>Date of Electronic Publication: </i>2022 Mar 29.
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        Value: 10.1021/acs.jmedchem.1c02048
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      – Code: eng
        Text: English
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              Text: 2022 Apr 14
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