Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells.

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Title: Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells.
Authors: Hosfield DJ; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Weber S; Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, Canada., Li NS; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Sauvage M; Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, Canada., Joiner CF; Department of Cancer Biology, Loyola University Chicago, Maywood, United States., Hancock GR; Department of Cancer Biology, Loyola University Chicago, Maywood, United States., Sullivan EA; Department of Cancer Biology, Loyola University Chicago, Maywood, United States., Ndukwe E; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Han R; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Cush S; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Lainé M; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Mader SC; Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, Canada., Greene GL; Ben May Department for Cancer Research, University of Chicago, Chicago, United States., Fanning SW; Department of Cancer Biology, Loyola University Chicago, Maywood, United States.
Source: ELife [Elife] 2022 May 16; Vol. 11. Date of Electronic Publication: 2022 May 16.
Publication Type: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, Non-U.S. Gov't
Journal Info: Publisher: eLife Sciences Publications, Ltd Country of Publication: England NLM ID: 101579614 Publication Model: Electronic Cited Medium: Internet ISSN: 2050-084X (Electronic) Linking ISSN: 2050084X NLM ISO Abbreviation: Elife Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells.
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  Data: <searchLink fieldCode="AU" term="%22Hosfield+DJ%22">Hosfield DJ</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Weber+S%22">Weber S</searchLink>; Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, Canada.<br /><searchLink fieldCode="AU" term="%22Li+NS%22">Li NS</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Sauvage+M%22">Sauvage M</searchLink>; Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, Canada.<br /><searchLink fieldCode="AU" term="%22Joiner+CF%22">Joiner CF</searchLink>; Department of Cancer Biology, Loyola University Chicago, Maywood, United States.<br /><searchLink fieldCode="AU" term="%22Hancock+GR%22">Hancock GR</searchLink>; Department of Cancer Biology, Loyola University Chicago, Maywood, United States.<br /><searchLink fieldCode="AU" term="%22Sullivan+EA%22">Sullivan EA</searchLink>; Department of Cancer Biology, Loyola University Chicago, Maywood, United States.<br /><searchLink fieldCode="AU" term="%22Ndukwe+E%22">Ndukwe E</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Han+R%22">Han R</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Cush+S%22">Cush S</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Lainé+M%22">Lainé M</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Mader+SC%22">Mader SC</searchLink>; Institute for Research in Immunology and Cancer, Université de Montréal, Montréal, Canada.<br /><searchLink fieldCode="AU" term="%22Greene+GL%22">Greene GL</searchLink>; Ben May Department for Cancer Research, University of Chicago, Chicago, United States.<br /><searchLink fieldCode="AU" term="%22Fanning+SW%22">Fanning SW</searchLink>; Department of Cancer Biology, Loyola University Chicago, Maywood, United States.
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  Data: <searchLink fieldCode="JN" term="%22101579614%22">ELife</searchLink> [Elife] 2022 May 16; Vol. 11. <i>Date of Electronic Publication: </i>2022 May 16.
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  Data: Journal Article; Research Support, U.S. Gov't, Non-P.H.S.; Research Support, Non-U.S. Gov't
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22eLife+Sciences+Publications%2C+Ltd%22">eLife Sciences Publications, Ltd </searchLink><i>Country of Publication: </i>England <i>NLM ID: </i>101579614 <i>Publication Model: </i>Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>2050-084X (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%222050084X%22">2050084X </searchLink><i>NLM ISO Abbreviation: </i>Elife <i>Subsets: </i>MEDLINE
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