Thiazole-based SARS-CoV-2 protease (COV Mpro ) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations.
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| Title: | Thiazole-based SARS-CoV-2 protease (COV Mpro ) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations. |
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| Authors: | Elsayed RW; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., Sabry MA; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., El-Subbagh HI; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., Bayoumi SM; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., El-Sayed SM; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt. |
| Source: | Archiv der Pharmazie [Arch Pharm (Weinheim)] 2022 Sep; Vol. 355 (9), pp. e2200121. Date of Electronic Publication: 2022 May 23. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 35607750 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Thiazole-based SARS-CoV-2 protease (COV M<superscript>pro</superscript> ) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Elsayed+RW%22">Elsayed RW</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.<br /><searchLink fieldCode="AU" term="%22Sabry+MA%22">Sabry MA</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.<br /><searchLink fieldCode="AU" term="%22El-Subbagh+HI%22">El-Subbagh HI</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.<br /><searchLink fieldCode="AU" term="%22Bayoumi+SM%22">Bayoumi SM</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.<br /><searchLink fieldCode="AU" term="%22El-Sayed+SM%22">El-Sayed SM</searchLink>; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%220330167%22">Archiv der Pharmazie</searchLink> [Arch Pharm (Weinheim)] 2022 Sep; Vol. 355 (9), pp. e2200121. <i>Date of Electronic Publication: </i>2022 May 23. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Wiley-VCH+Verlag+GmbH+%26+Co%2E+KGaA%22">Wiley-VCH Verlag GmbH & Co. KGaA </searchLink><i>Country of Publication: </i>Germany <i>NLM ID: </i>0330167 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1521-4184 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2203656233%22">03656233 </searchLink><i>NLM ISO Abbreviation: </i>Arch Pharm (Weinheim) <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=35607750 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1002/ardp.202200121 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: e2200121 Titles: – TitleFull: Thiazole-based SARS-CoV-2 protease (COV Mpro ) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Elsayed RW – PersonEntity: Name: NameFull: Sabry MA – PersonEntity: Name: NameFull: El-Subbagh HI – PersonEntity: Name: NameFull: Bayoumi SM – PersonEntity: Name: NameFull: El-Sayed SM IsPartOfRelationships: – BibEntity: Dates: – D: 01 M: 09 Text: 2022 Sep Type: published Y: 2022 Identifiers: – Type: issn-electronic Value: 1521-4184 Numbering: – Type: volume Value: 355 – Type: issue Value: 9 Titles: – TitleFull: Archiv der Pharmazie Type: main |
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