Quinazoline-based human phosphodiesterase 5 inhibitors exhibited a selective vasorelaxant effect on rat isolated pulmonary arteries involving NO-sGC-cGMP pathway and calcium inhibitory effects.

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Title: Quinazoline-based human phosphodiesterase 5 inhibitors exhibited a selective vasorelaxant effect on rat isolated pulmonary arteries involving NO-sGC-cGMP pathway and calcium inhibitory effects.
Authors: Chatturong U; Department of Physiology, Faculty of Medical Science and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France., Martin H; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France., Totoson P; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France., Ingkaninan K; Department of Pharmaceutical Chemistry and Pharmacognosy, Faculty of Pharmaceutical Sciences and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand., Temkitthawon P; Department of Pharmaceutical Chemistry and Pharmacognosy, Faculty of Pharmaceutical Sciences and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand., Sermsenaphorn S; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand., Somarin T; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand., Konsue A; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand., Gleeson MP; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand., Demougeot C; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France., Chootip K; Department of Physiology, Faculty of Medical Science and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand. Electronic address: krongkarnc@nu.ac.th.
Source: Vascular pharmacology [Vascul Pharmacol] 2022 Dec; Vol. 147, pp. 107111. Date of Electronic Publication: 2022 Sep 24.
Publication Type: Journal Article; Research Support, Non-U.S. Gov't
Journal Info: Publisher: Elsevier Science Country of Publication: United States NLM ID: 101130615 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1879-3649 (Electronic) Linking ISSN: 15371891 NLM ISO Abbreviation: Vascul Pharmacol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Quinazoline-based human phosphodiesterase 5 inhibitors exhibited a selective vasorelaxant effect on rat isolated pulmonary arteries involving NO-sGC-cGMP pathway and calcium inhibitory effects.
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  Data: <searchLink fieldCode="AU" term="%22Chatturong+U%22">Chatturong U</searchLink>; Department of Physiology, Faculty of Medical Science and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France.<br /><searchLink fieldCode="AU" term="%22Martin+H%22">Martin H</searchLink>; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France.<br /><searchLink fieldCode="AU" term="%22Totoson+P%22">Totoson P</searchLink>; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France.<br /><searchLink fieldCode="AU" term="%22Ingkaninan+K%22">Ingkaninan K</searchLink>; Department of Pharmaceutical Chemistry and Pharmacognosy, Faculty of Pharmaceutical Sciences and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand.<br /><searchLink fieldCode="AU" term="%22Temkitthawon+P%22">Temkitthawon P</searchLink>; Department of Pharmaceutical Chemistry and Pharmacognosy, Faculty of Pharmaceutical Sciences and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand.<br /><searchLink fieldCode="AU" term="%22Sermsenaphorn+S%22">Sermsenaphorn S</searchLink>; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand.<br /><searchLink fieldCode="AU" term="%22Somarin+T%22">Somarin T</searchLink>; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand.<br /><searchLink fieldCode="AU" term="%22Konsue+A%22">Konsue A</searchLink>; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand.<br /><searchLink fieldCode="AU" term="%22Gleeson+MP%22">Gleeson MP</searchLink>; Department of Biomedical Engineering, Faculty of Engineering, King Mongkut's Institute of Technology, Ladkrabang, Bangkok 10520, Thailand.<br /><searchLink fieldCode="AU" term="%22Demougeot+C%22">Demougeot C</searchLink>; PEPITE EA4267, Université Bourgogne Franche-Comté, Besançon 25030, France.<br /><searchLink fieldCode="AU" term="%22Chootip+K%22">Chootip K</searchLink>; Department of Physiology, Faculty of Medical Science and Center of Excellence for Innovation in Chemistry, Naresuan University, Phitsanulok 65000, Thailand. Electronic address: krongkarnc@nu.ac.th.
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  Data: <searchLink fieldCode="JN" term="%22101130615%22">Vascular pharmacology</searchLink> [Vascul Pharmacol] 2022 Dec; Vol. 147, pp. 107111. <i>Date of Electronic Publication: </i>2022 Sep 24.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier+Science%22">Elsevier Science </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101130615 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1879-3649 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2215371891%22">15371891 </searchLink><i>NLM ISO Abbreviation: </i>Vascul Pharmacol <i>Subsets: </i>MEDLINE
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        Value: 10.1016/j.vph.2022.107111
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              Text: 2022 Dec
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