Structural basis of synthetic agonist activation of the nuclear receptor REV-ERB.

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Title: Structural basis of synthetic agonist activation of the nuclear receptor REV-ERB.
Authors: Murray MH; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, St. Louis, MO, 63104, USA.; Center for Clinical Pharmacology, Washington University School of Medicine, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA., Valfort AC; University of Florida Genetics Institute, Gainesville, FL, 32610, USA., Koelblen T; University of Florida Genetics Institute, Gainesville, FL, 32610, USA., Ronin C; NovAliX SAS, Strasbourg, France., Ciesielski F; NovAliX SAS, Strasbourg, France., Chatterjee A; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, St. Louis, MO, 63104, USA., Veerakanellore GB; Center for Clinical Pharmacology, Washington University School of Medicine, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA.; Department of Pharmaceutical and Administrative Sciences, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA., Elgendy B; Center for Clinical Pharmacology, Washington University School of Medicine, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA.; Department of Pharmaceutical and Administrative Sciences, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA., Walker JK; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, St. Louis, MO, 63104, USA., Hegazy L; Center for Clinical Pharmacology, Washington University School of Medicine, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA. Lamees.Hegazy@uhsp.edu.; Department of Pharmaceutical and Administrative Sciences, University of Health Sciences & Pharmacy, St. Louis, MO, 63110, USA. Lamees.Hegazy@uhsp.edu., Burris TP; University of Florida Genetics Institute, Gainesville, FL, 32610, USA. burris.thomas@ufl.edu.
Source: Nature communications [Nat Commun] 2022 Nov 21; Vol. 13 (1), pp. 7131. Date of Electronic Publication: 2022 Nov 21.
Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, U.S. Gov't, Non-P.H.S.
Journal Info: Publisher: Nature Pub. Group Country of Publication: England NLM ID: 101528555 Publication Model: Electronic Cited Medium: Internet ISSN: 2041-1723 (Electronic) Linking ISSN: 20411723 NLM ISO Abbreviation: Nat Commun Subsets: MEDLINE
Database: MEDLINE Ultimate
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ISSN:2041-1723
DOI:10.1038/s41467-022-34892-4