Chemical Biology Approaches Confirm MCT4 as the Therapeutic Target of a Cellular Optimized Hit.

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Title: Chemical Biology Approaches Confirm MCT4 as the Therapeutic Target of a Cellular Optimized Hit.
Authors: Kawatkar A; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Clark RA; Discovery Sciences, R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Hopcroft L; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Roaquin DA; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Tomlinson R; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Zuhl AM; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Lamont GM; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Kettle JG; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Critchlow SE; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Castaldi MP; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Goldberg FW; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Zhang AX; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.
Source: ACS chemical biology [ACS Chem Biol] 2023 Feb 17; Vol. 18 (2), pp. 296-303. Date of Electronic Publication: 2023 Jan 05.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
Description
ISSN:1554-8937
DOI:10.1021/acschembio.2c00666