Chemical Biology Approaches Confirm MCT4 as the Therapeutic Target of a Cellular Optimized Hit.

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Title: Chemical Biology Approaches Confirm MCT4 as the Therapeutic Target of a Cellular Optimized Hit.
Authors: Kawatkar A; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Clark RA; Discovery Sciences, R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Hopcroft L; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Roaquin DA; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Tomlinson R; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Zuhl AM; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Lamont GM; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Kettle JG; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Critchlow SE; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Castaldi MP; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States., Goldberg FW; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K., Zhang AX; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.
Source: ACS chemical biology [ACS Chem Biol] 2023 Feb 17; Vol. 18 (2), pp. 296-303. Date of Electronic Publication: 2023 Jan 05.
Publication Type: Journal Article
Journal Info: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101282906 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1554-8937 (Electronic) Linking ISSN: 15548929 NLM ISO Abbreviation: ACS Chem Biol Subsets: MEDLINE
Database: MEDLINE Ultimate
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  Data: Chemical Biology Approaches Confirm MCT4 as the Therapeutic Target of a Cellular Optimized Hit.
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  Data: <searchLink fieldCode="AU" term="%22Kawatkar+A%22">Kawatkar A</searchLink>; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.<br /><searchLink fieldCode="AU" term="%22Clark+RA%22">Clark RA</searchLink>; Discovery Sciences, R&D, AstraZeneca, CambridgeCB2 0AA, U.K.<br /><searchLink fieldCode="AU" term="%22Hopcroft+L%22">Hopcroft L</searchLink>; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K.<br /><searchLink fieldCode="AU" term="%22Roaquin+DA%22">Roaquin DA</searchLink>; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.<br /><searchLink fieldCode="AU" term="%22Tomlinson+R%22">Tomlinson R</searchLink>; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.<br /><searchLink fieldCode="AU" term="%22Zuhl+AM%22">Zuhl AM</searchLink>; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.<br /><searchLink fieldCode="AU" term="%22Lamont+GM%22">Lamont GM</searchLink>; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K.<br /><searchLink fieldCode="AU" term="%22Kettle+JG%22">Kettle JG</searchLink>; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K.<br /><searchLink fieldCode="AU" term="%22Critchlow+SE%22">Critchlow SE</searchLink>; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K.<br /><searchLink fieldCode="AU" term="%22Castaldi+MP%22">Castaldi MP</searchLink>; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.<br /><searchLink fieldCode="AU" term="%22Goldberg+FW%22">Goldberg FW</searchLink>; Oncology R&D, AstraZeneca, CambridgeCB2 0AA, U.K.<br /><searchLink fieldCode="AU" term="%22Zhang+AX%22">Zhang AX</searchLink>; Discovery Sciences, R&D, AstraZeneca, Waltham, Massachusetts02451, United States.
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  Data: <searchLink fieldCode="JN" term="%22101282906%22">ACS chemical biology</searchLink> [ACS Chem Biol] 2023 Feb 17; Vol. 18 (2), pp. 296-303. <i>Date of Electronic Publication: </i>2023 Jan 05.
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  Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101282906 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1554-8937 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2215548929%22">15548929 </searchLink><i>NLM ISO Abbreviation: </i>ACS Chem Biol <i>Subsets: </i>MEDLINE
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        Value: 10.1021/acschembio.2c00666
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              Text: 2023 Feb 17
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