Discovery of Paltusotine (CRN00808), a Potent, Selective, and Orally Bioavailable Non-peptide SST2 Agonist.
Saved in:
| Title: | Discovery of Paltusotine (CRN00808), a Potent, Selective, and Orally Bioavailable Non-peptide SST2 Agonist. |
|---|---|
| Authors: | Zhao J; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Wang S; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Markison S; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Kim SH; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Han S; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Chen M; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Kusnetzow AK; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Rico-Bautista E; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Johns M; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Luo R; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Struthers RS; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Madan A; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Zhu Y; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States., Betz SF; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States. |
| Source: | ACS medicinal chemistry letters [ACS Med Chem Lett] 2022 Dec 10; Vol. 14 (1), pp. 66-74. Date of Electronic Publication: 2022 Dec 10 (Print Publication: 2023). |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: American Chemical Society Country of Publication: United States NLM ID: 101521073 Publication Model: eCollection Cited Medium: Print ISSN: 1948-5875 (Print) Linking ISSN: 19485875 NLM ISO Abbreviation: ACS Med Chem Lett Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
|---|---|
| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 36655128 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
| IllustrationInfo | |
| Items | – Name: Title Label: Title Group: Ti Data: Discovery of Paltusotine (CRN00808), a Potent, Selective, and Orally Bioavailable Non-peptide SST2 Agonist. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Zhao+J%22">Zhao J</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Wang+S%22">Wang S</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Markison+S%22">Markison S</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Kim+SH%22">Kim SH</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Han+S%22">Han S</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Chen+M%22">Chen M</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Kusnetzow+AK%22">Kusnetzow AK</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Rico-Bautista+E%22">Rico-Bautista E</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Johns+M%22">Johns M</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Luo+R%22">Luo R</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Struthers+RS%22">Struthers RS</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Madan+A%22">Madan A</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Zhu+Y%22">Zhu Y</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States.<br /><searchLink fieldCode="AU" term="%22Betz+SF%22">Betz SF</searchLink>; Crinetics Pharmaceuticals, Inc., 10222 Barnes Canyon Road, Building #2, San Diego, California 92121, United States. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%22101521073%22">ACS medicinal chemistry letters</searchLink> [ACS Med Chem Lett] 2022 Dec 10; Vol. 14 (1), pp. 66-74. <i>Date of Electronic Publication: </i>2022 Dec 10 (<i>Print Publication: </i>2023). – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22American+Chemical+Society%22">American Chemical Society </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>101521073 <i>Publication Model: </i>eCollection <i>Cited Medium: </i>Print <i>ISSN: </i>1948-5875 (Print) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2219485875%22">19485875 </searchLink><i>NLM ISO Abbreviation: </i>ACS Med Chem Lett <i>Subsets: </i>PubMed not MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=36655128 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1021/acsmedchemlett.2c00431 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 66 Titles: – TitleFull: Discovery of Paltusotine (CRN00808), a Potent, Selective, and Orally Bioavailable Non-peptide SST2 Agonist. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Zhao J – PersonEntity: Name: NameFull: Wang S – PersonEntity: Name: NameFull: Markison S – PersonEntity: Name: NameFull: Kim SH – PersonEntity: Name: NameFull: Han S – PersonEntity: Name: NameFull: Chen M – PersonEntity: Name: NameFull: Kusnetzow AK – PersonEntity: Name: NameFull: Rico-Bautista E – PersonEntity: Name: NameFull: Johns M – PersonEntity: Name: NameFull: Luo R – PersonEntity: Name: NameFull: Struthers RS – PersonEntity: Name: NameFull: Madan A – PersonEntity: Name: NameFull: Zhu Y – PersonEntity: Name: NameFull: Betz SF IsPartOfRelationships: – BibEntity: Dates: – D: 10 M: 12 Text: 2022 Dec 10 Type: published Y: 2022 Identifiers: – Type: issn-print Value: 1948-5875 Numbering: – Type: volume Value: 14 – Type: issue Value: 1 Titles: – TitleFull: ACS medicinal chemistry letters Type: main |
| ResultId | 1 |
