Comparative analysis of drug-like EP300/CREBBP acetyltransferase inhibitors.

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Title: Comparative analysis of drug-like EP300/CREBBP acetyltransferase inhibitors.
Authors: Crawford MC; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Tripu DR; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Barritt SA; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA, USA., Jing Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Gallimore D; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Kales SC; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Bhanu NV; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, MO, USA., Xiong Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Fang Y; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Butler KAT; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., LeClair CA; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Coussens NP; Molecular Pharmacology Laboratories, Applied and Developmental Research Directorate, Frederick National Laboratory for Cancer Research, Frederick, MD, USA., Simeonov A; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Garcia BA; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, MO, USA., Dibble CC; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA, USA., Meier JL; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA, USA.
Source: BioRxiv : the preprint server for biology [bioRxiv] 2023 May 16. Date of Electronic Publication: 2023 May 16.
Publication Type: Preprint; Journal Article
Journal Info: Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE
Database: MEDLINE Ultimate
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  Data: Comparative analysis of drug-like EP300/CREBBP acetyltransferase inhibitors.
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