Comparative analysis of drug-like EP300/CREBBP acetyltransferase inhibitors.
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| Title: | Comparative analysis of drug-like EP300/CREBBP acetyltransferase inhibitors. |
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| Authors: | Crawford MC; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Tripu DR; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Barritt SA; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA, USA., Jing Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Gallimore D; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Kales SC; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Bhanu NV; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, MO, USA., Xiong Y; Chemical Biology Laboratory, National Cancer Institute, Frederick, MD, USA., Fang Y; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Butler KAT; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., LeClair CA; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Coussens NP; Molecular Pharmacology Laboratories, Applied and Developmental Research Directorate, Frederick National Laboratory for Cancer Research, Frederick, MD, USA., Simeonov A; National Center for Advancing Translational Sciences, National Institutes of Health, Rockville, MD, USA., Garcia BA; Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, MO, USA., Dibble CC; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA, USA., Meier JL; Department of Pathology, Cancer Research Institute, Beth Israel Deaconess Medical Center, Harvard Medical School, Boston, MA, USA. |
| Source: | BioRxiv : the preprint server for biology [bioRxiv] 2023 May 16. Date of Electronic Publication: 2023 May 16. |
| Publication Type: | Preprint; Journal Article |
| Journal Info: | Country of Publication: United States NLM ID: 101680187 Publication Model: Electronic Cited Medium: Internet ISSN: 2692-8205 (Electronic) Linking ISSN: 26928205 NLM ISO Abbreviation: bioRxiv Subsets: PubMed not MEDLINE |
| Database: | MEDLINE Ultimate |
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