Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915.
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| Title: | Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915. |
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| Authors: | Hampton CS; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Sitaula S; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States., Billon C; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States., Haynes K; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Avdagic A; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Wanninayake U; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Adeyemi CM; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Chatterjee A; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Griffett K; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States., Banerjee S; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Burris SL; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States., Schoepke E; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Boehm T; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Bess A; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., de Vera IMS; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States., Burris TP; University of Florida Genetics Institute, Gainesville, FL, 32310, USA., Walker JK; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States; Institute for Translational Neuroscience, Saint Louis University, St. Louis MO, 63110, United States. Electronic address: john.walker@health.slu.edu. |
| Source: | European journal of medicinal chemistry [Eur J Med Chem] 2023 Oct 05; Vol. 258, pp. 115582. Date of Electronic Publication: 2023 Jun 25. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 37421886 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Hampton+CS%22">Hampton CS</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Sitaula+S%22">Sitaula S</searchLink>; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States.<br /><searchLink fieldCode="AU" term="%22Billon+C%22">Billon C</searchLink>; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States.<br /><searchLink fieldCode="AU" term="%22Haynes+K%22">Haynes K</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Avdagic+A%22">Avdagic A</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Wanninayake+U%22">Wanninayake U</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Adeyemi+CM%22">Adeyemi CM</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Chatterjee+A%22">Chatterjee A</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Griffett+K%22">Griffett K</searchLink>; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States.<br /><searchLink fieldCode="AU" term="%22Banerjee+S%22">Banerjee S</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Burris+SL%22">Burris SL</searchLink>; Center for Clinical Pharmacology, St. Louis College of Pharmacy, Saint Louis, Missouri, 63110, United States.<br /><searchLink fieldCode="AU" term="%22Schoepke+E%22">Schoepke E</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Boehm+T%22">Boehm T</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Bess+A%22">Bess A</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22de+Vera+IMS%22">de Vera IMS</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States.<br /><searchLink fieldCode="AU" term="%22Burris+TP%22">Burris TP</searchLink>; University of Florida Genetics Institute, Gainesville, FL, 32310, USA.<br /><searchLink fieldCode="AU" term="%22Walker+JK%22">Walker JK</searchLink>; Department of Pharmacology and Physiology, Saint Louis University School of Medicine, Saint Louis, Missouri, 63104, United States; Institute for Translational Neuroscience, Saint Louis University, St. Louis MO, 63110, United States. Electronic address: john.walker@health.slu.edu. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%220420510%22">European journal of medicinal chemistry</searchLink> [Eur J Med Chem] 2023 Oct 05; Vol. 258, pp. 115582. <i>Date of Electronic Publication: </i>2023 Jun 25. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Editions+Scientifiques+Elsevier%22">Editions Scientifiques Elsevier </searchLink><i>Country of Publication: </i>France <i>NLM ID: </i>0420510 <i>Publication Model: </i>Print-Electronic <i>Cited Medium: </i>Internet <i>ISSN: </i>1768-3254 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2202235234%22">02235234 </searchLink><i>NLM ISO Abbreviation: </i>Eur J Med Chem <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=37421886 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1016/j.ejmech.2023.115582 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 115582 Titles: – TitleFull: Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Hampton CS – PersonEntity: Name: NameFull: Sitaula S – PersonEntity: Name: NameFull: Billon C – PersonEntity: Name: NameFull: Haynes K – PersonEntity: Name: NameFull: Avdagic A – PersonEntity: Name: NameFull: Wanninayake U – PersonEntity: Name: NameFull: Adeyemi CM – PersonEntity: Name: NameFull: Chatterjee A – PersonEntity: Name: NameFull: Griffett K – PersonEntity: Name: NameFull: Banerjee S – PersonEntity: Name: NameFull: Burris SL – PersonEntity: Name: NameFull: Schoepke E – PersonEntity: Name: NameFull: Boehm T – PersonEntity: Name: NameFull: Bess A – PersonEntity: Name: NameFull: de Vera IMS – PersonEntity: Name: NameFull: Burris TP – PersonEntity: Name: NameFull: Walker JK IsPartOfRelationships: – BibEntity: Dates: – D: 05 M: 10 Text: 2023 Oct 05 Type: published Y: 2023 Identifiers: – Type: issn-electronic Value: 1768-3254 Numbering: – Type: volume Value: 258 Titles: – TitleFull: European journal of medicinal chemistry Type: main |
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