Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors.
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| Title: | Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors. |
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| Authors: | Mobbs JI; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia., Black KA; Structural Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, Australia.; Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia.; Department of Biochemistry and Pharmacology, University of Melbourne, Melbourne, VIC, Australia., Tran M; Department of Chemistry and Biochemistry, University of California, Santa Cruz, Santa Cruz, CA., Burger WAC; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; Structural Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, Australia.; Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia.; Department of Biochemistry and Pharmacology, University of Melbourne, Melbourne, VIC, Australia., Venugopal H; Ramaciotti Centre for Cryo-Electron Microscopy, Monash University, Clayton, VIC, Australia., Holman TR; Department of Chemistry and Biochemistry, University of California, Santa Cruz, Santa Cruz, CA., Holinstat M; Department of Pharmacology, University of Michigan, Ann Arbor, MI.; Division of Cardiovascular Medicine, Department of Internal Medicine, University of Michigan, Ann Arbor, MI., Thal DM; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia., Glukhova A; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; Structural Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, Australia.; Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia.; Department of Biochemistry and Pharmacology, University of Melbourne, Melbourne, VIC, Australia. |
| Source: | Blood [Blood] 2023 Oct 05; Vol. 142 (14), pp. 1233-1242. |
| Publication Type: | Journal Article |
| Journal Info: | Publisher: Elsevier Country of Publication: United States NLM ID: 7603509 Publication Model: Print Cited Medium: Internet ISSN: 1528-0020 (Electronic) Linking ISSN: 00064971 NLM ISO Abbreviation: Blood Subsets: MEDLINE |
| Database: | MEDLINE Ultimate |
| FullText | Text: Availability: 0 |
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| Header | DbId: mdl DbLabel: MEDLINE Ultimate An: 37506345 AccessLevel: 2 PubType: Academic Journal PubTypeId: academicJournal PreciseRelevancyScore: 0 |
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| Items | – Name: Title Label: Title Group: Ti Data: Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors. – Name: Author Label: Authors Group: Au Data: <searchLink fieldCode="AU" term="%22Mobbs+JI%22">Mobbs JI</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.<br /><searchLink fieldCode="AU" term="%22Black+KA%22">Black KA</searchLink>; Structural Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, Australia.; Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia.; Department of Biochemistry and Pharmacology, University of Melbourne, Melbourne, VIC, Australia.<br /><searchLink fieldCode="AU" term="%22Tran+M%22">Tran M</searchLink>; Department of Chemistry and Biochemistry, University of California, Santa Cruz, Santa Cruz, CA.<br /><searchLink fieldCode="AU" term="%22Burger+WAC%22">Burger WAC</searchLink>; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; Structural Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, Australia.; Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia.; Department of Biochemistry and Pharmacology, University of Melbourne, Melbourne, VIC, Australia.<br /><searchLink fieldCode="AU" term="%22Venugopal+H%22">Venugopal H</searchLink>; Ramaciotti Centre for Cryo-Electron Microscopy, Monash University, Clayton, VIC, Australia.<br /><searchLink fieldCode="AU" term="%22Holman+TR%22">Holman TR</searchLink>; Department of Chemistry and Biochemistry, University of California, Santa Cruz, Santa Cruz, CA.<br /><searchLink fieldCode="AU" term="%22Holinstat+M%22">Holinstat M</searchLink>; Department of Pharmacology, University of Michigan, Ann Arbor, MI.; Division of Cardiovascular Medicine, Department of Internal Medicine, University of Michigan, Ann Arbor, MI.<br /><searchLink fieldCode="AU" term="%22Thal+DM%22">Thal DM</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.<br /><searchLink fieldCode="AU" term="%22Glukhova+A%22">Glukhova A</searchLink>; Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; ARC Centre for Cryo-Electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.; Structural Biology Division, Walter and Eliza Hall Institute of Medical Research, Parkville, VIC, Australia.; Department of Medical Biology, University of Melbourne, Melbourne, VIC, Australia.; Department of Biochemistry and Pharmacology, University of Melbourne, Melbourne, VIC, Australia. – Name: TitleSource Label: Source Group: Src Data: <searchLink fieldCode="JN" term="%227603509%22">Blood</searchLink> [Blood] 2023 Oct 05; Vol. 142 (14), pp. 1233-1242. – Name: TypePub Label: Publication Type Group: TypPub Data: Journal Article – Name: TitleSource Label: Journal Info Group: Src Data: <i>Publisher: </i><searchLink fieldCode="PB" term="%22Elsevier%22">Elsevier </searchLink><i>Country of Publication: </i>United States <i>NLM ID: </i>7603509 <i>Publication Model: </i>Print <i>Cited Medium: </i>Internet <i>ISSN: </i>1528-0020 (Electronic) <i>Linking ISSN: </i><searchLink fieldCode="IS" term="%2200064971%22">00064971 </searchLink><i>NLM ISO Abbreviation: </i>Blood <i>Subsets: </i>MEDLINE |
| PLink | https://search.ebscohost.com/login.aspx?direct=true&site=eds-live&db=mdl&AN=37506345 |
| RecordInfo | BibRecord: BibEntity: Identifiers: – Type: doi Value: 10.1182/blood.2023020441 Languages: – Code: eng Text: English PhysicalDescription: Pagination: StartPage: 1233 Titles: – TitleFull: Cryo-EM structures of human arachidonate 12S-lipoxygenase bound to endogenous and exogenous inhibitors. Type: main BibRelationships: HasContributorRelationships: – PersonEntity: Name: NameFull: Mobbs JI – PersonEntity: Name: NameFull: Black KA – PersonEntity: Name: NameFull: Tran M – PersonEntity: Name: NameFull: Burger WAC – PersonEntity: Name: NameFull: Venugopal H – PersonEntity: Name: NameFull: Holman TR – PersonEntity: Name: NameFull: Holinstat M – PersonEntity: Name: NameFull: Thal DM – PersonEntity: Name: NameFull: Glukhova A IsPartOfRelationships: – BibEntity: Dates: – D: 05 M: 10 Text: 2023 Oct 05 Type: published Y: 2023 Identifiers: – Type: issn-electronic Value: 1528-0020 Numbering: – Type: volume Value: 142 – Type: issue Value: 14 Titles: – TitleFull: Blood Type: main |
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